SCHEMBL22453875

SCHEMBL22453875

CC(=N)c1cc(NC(=O)c2c(C)cc3c(C)ncn3c2C)ccc1N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.46
LCK P06239 2/20 0.33
KDR P35968 2/20 0.33
SMN1; SMN2 Q16637 5/20 0.33
RAB9A P51151 5/20 0.33
NPC1 O15118 4/20 0.33
LMNA P02545 2/20 0.33
AURKA O14965 1/20 0.32
AURKB Q96GD4 1/20 0.32
HTT P42858 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 2/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32
ALDH1A1 P00352 1/20 0.32
FADS1 O60427 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
BTK Q06187 1/20 0.31
MAPK14 Q16539 1/20 0.31
MEN1 O00255 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453946 0.84 LRRK2 (0.35) LRRK2LCKSMN1; SMN2RAB9ANPC1
SCHEMBL22453185 0.77 LRRK2 (0.46) LRRK2SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL22453793 0.75 LRRK2 (0.46) LRRK2SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL22452978 0.74 LRRK2 (0.51) LRRK2SMN1; SMN2RAB9ANPC1LMNA
SCHEMBL22453874 0.74 LRRK2 (0.43) LRRK2
SCHEMBL22453892 0.71 LRRK2 (0.55) LRRK2SMN1; SMN2RAB9ANPC1ALDH1A1
SCHEMBL22453216 0.68 LRRK2 (0.47) LRRK2LCKKDRSMN1; SMN2RAB9A
SCHEMBL22445872 0.68 SMN1; SMN2 (0.39) SMN1; SMN2LMNATP53MAPTALDH1A1
SCHEMBL22452996 0.68 LRRK2 (0.50) LRRK2RAB9ANPC1LMNAMAPT
SCHEMBL22453384 0.67 LRRK2 (0.50) LRRK2SMN1; SMN2RAB9AALDH1A1FADS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020191261-A1 INDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2020-09-24 WO disclosed