SCHEMBL22453384

SCHEMBL22453384

CNc1cc(C)c(C(=O)Nc2ccc(N)c(C(C)=N)c2)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.50
PRKCI P41743 1/20 0.43
HDAC1 Q13547 5/20 0.39
FADS1 O60427 3/20 0.38
ALDH1A1 P00352 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
F2 P00734 3/20 0.38
F10 P00742 3/20 0.38
PLAU P00749 3/20 0.38
PLAT P00750 3/20 0.38
PLG P00747 2/20 0.38
KLK1 P06870 1/20 0.38
KLK5 Q9Y337 1/20 0.38
KDM4E B2RXH2 1/20 0.37
RAB9A P51151 1/20 0.37
BRAF P15056 2/20 0.37
HDAC8 Q9BY41 2/20 0.37
HDAC6 Q9UBN7 2/20 0.37
HDAC3 O15379 1/20 0.37
HDAC4 P56524 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453892 0.89 LRRK2 (0.55) LRRK2HDAC1FADS1ALDH1A1SMN1; SMN2
SCHEMBL22453421 0.77 LRRK2 (0.43) LRRK2HDAC1FADS1ALDH1A1SMN1; SMN2
SCHEMBL22453429 0.77 LRRK2 (0.42) LRRK2PRKCIHDAC1KDM4ERAB9A
SCHEMBL22452996 0.77 LRRK2 (0.50) LRRK2HDAC1F2PLAUPLAT
SCHEMBL22889931 0.76 LRRK2 (0.59) LRRK2ALDH1A1SMN1; SMN2F2F10
SCHEMBL22453342 0.74 LRRK2 (0.46) LRRK2HDAC1FADS1BRAFHDAC8
SCHEMBL22452978 0.74 LRRK2 (0.51) LRRK2FADS1ALDH1A1SMN1; SMN2F2
SCHEMBL22454024 0.73 KMT2A (0.48) HDAC1ALDH1A1SMN1; SMN2F2F10
SCHEMBL22452969 0.72 LRRK2 (0.48) LRRK2HDAC1FADS1SMN1; SMN2RAB9A
SCHEMBL22065324 0.70 FADS1 (0.54) HDAC1FADS1ALDH1A1SMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020191261-A1 INDAZOLES AS LRRK2 INHIBITORS E-SCAPE BIO, INC. (US) 2020-09-24 WO disclosed