SCHEMBL22453584

SCHEMBL22453584

CCOC(=O)c1cccc(Nc2ccc(C(=O)Nc3ccc(C4CCCCC4)cc3)cc2C)n1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.44
HDAC11 Q96DB2 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
DEGS1 O15121 1/20 0.44
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
NAMPT P43490 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
GAA P10253 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22453296 0.89 HDAC3 (0.47) HDAC3HDAC11HDAC8HDAC6DEGS1
SCHEMBL22452937 0.83 DHODH (0.40) TP53MAPTGAA
SCHEMBL22453576 0.83 CYP1A2 (0.40) MAPTSMN1; SMN2NPC1
SCHEMBL22453719 0.77 CYP1A2 (0.37) MAPTSMN1; SMN2
SCHEMBL22453578 0.77 MAPT (0.42) MAPTSMN1; SMN2NPC1GAA
SCHEMBL22452936 0.77 NR1H4 (0.35) TP53MAPTSMN1; SMN2
SCHEMBL22452648 0.76 RAB9A (0.49) HDAC3HDAC11HDAC8HDAC6DEGS1
SCHEMBL22452774 0.74 MEN1 (0.52) HDAC3HDAC11HDAC8HDAC6DEGS1
SCHEMBL22453482 0.71 SMN1; SMN2 (0.53) HDAC3HDAC11HDAC8HDAC6DEGS1
SCHEMBL22452929 0.70 HDAC3 (0.62) HDAC3HDAC11HDAC8HDAC6DEGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed