SCHEMBL22453576

SCHEMBL22453576

CCOC(=O)c1cccc(Nc2ccc(N(C)c3ccc(C4CCCCC4)cc3)cc2C)n1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
KDM4C Q9H3R0 4/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
KDM6B O15054 2/20 0.36
KDM4E B2RXH2 3/20 0.35
NR1H4 Q96RI1 2/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
TSHR P16473 1/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALOX15 P16050 1/20 0.35
GRM5 P41594 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
NPC1 O15118 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22452936 0.89 NR1H4 (0.35) CYP1A2MEN1KMT2ANR1H4ALDH1A1
SCHEMBL22453719 0.88 CYP1A2 (0.37) CYP1A2KDM4CMEN1KMT2AKDM6B
SCHEMBL22452558 0.88 KDM4C (0.42) KDM4CMEN1KMT2AKDM6BKDM4E
SCHEMBL22453716 0.83 PDCD1 (0.36) CYP1A2KDM4CMEN1KMT2AKDM6B
SCHEMBL22453584 0.83 HDAC3 (0.44) MAPTSMN1; SMN2NPC1
SCHEMBL22453579 0.81 CYP1A2 (0.42) CYP1A2KDM4CKDM6BKDM4ELMNA
SCHEMBL22452937 0.81 DHODH (0.40) CYP1A2MEN1KMT2AALDH1A1MAPT
SCHEMBL22453585 0.81 CYP1A2 (0.38) CYP1A2MEN1KMT2AKDM4ENR1H4
SCHEMBL22453582 0.79 KDM4C (0.41) CYP1A2KDM4CMEN1KMT2AKDM4E
SCHEMBL22453086 0.78 SERPINE1 (0.35) KDM4CKMT2AKDM4ELMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed