SCHEMBL22453743

SCHEMBL22453743

Cc1cc(C(=O)O)ccc1Nc1ccc(C2CCCCC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.55
KMO O15229 1/20 0.49
KMT2A Q03164 4/20 0.48
ALDH1A1 P00352 4/20 0.48
MEN1 O00255 2/20 0.48
POLB P06746 1/20 0.48
SERPINE1 P05121 1/20 0.48
KDM4E B2RXH2 5/20 0.48
NPC1 O15118 3/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
GAA P10253 3/20 0.48
MAPT P10636 3/20 0.48
GFER P55789 1/20 0.48
HDAC8 Q9BY41 2/20 0.47
HDAC6 Q9UBN7 2/20 0.47
HDAC3 O15379 1/20 0.47
HDAC11 Q96DB2 1/20 0.47
DEGS1 O15121 1/20 0.47
HAO1 Q9UJM8 1/20 0.46
HDAC1 Q13547 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31003876 0.91 KMO (0.50) S1PR1KMOKMT2AALDH1A1MEN1
SCHEMBL22452774 0.88 MEN1 (0.52) S1PR1KMOKMT2AALDH1A1MEN1
SCHEMBL22453482 0.88 SMN1; SMN2 (0.53) S1PR1KMT2AALDH1A1MEN1SERPINE1
SCHEMBL28592246 0.84 KDM4E (0.49) S1PR1KMOKMT2AALDH1A1MEN1
SCHEMBL22453749 0.82 HDAC8 (0.57) KMOKMT2AALDH1A1MEN1POLB
SCHEMBL20400984 0.81 S1PR1 (0.49) S1PR1KMOKMT2AALDH1A1MEN1
SCHEMBL25053698 0.81 MAPT (0.49) KMT2AALDH1A1MEN1POLBNPC1
SCHEMBL22452648 0.78 RAB9A (0.49) KMT2AALDH1A1MEN1NPC1SMN1; SMN2
SCHEMBL25053696 0.78 MAPT (0.44) KMT2AALDH1A1MEN1NPC1SMN1; SMN2
SCHEMBL31003814 0.76 KMO (0.54) KMOKMT2AALDH1A1MEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020190774-A1 NOVEL SMALL MOLECULE INHIBITORS OF TEAD TRANSCRIPTION FACTORS THE GENERAL HOSPITAL CORPORATION (US) 2020-09-24 WO disclosed