SCHEMBL22463151

SCHEMBL22463151

Fc1cc[c]c(-c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AHR P35869 5/20 0.46
CYP1B1 Q16678 1/20 0.41
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
NOTUM Q6P988 2/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
PTGS2 P35354 1/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
GAA P10253 1/20 0.33
PKM P14618 1/20 0.33
ALOX12 P18054 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
KMO O15229 3/20 0.33
TP53 P04637 1/20 0.32
PPP1CA P62136 1/20 0.32
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9804988 0.81 AHR (0.50) AHRCYP1B1NPC1RAB9ANOTUM
SCHEMBL436469 0.81 NOTUM (0.38) AHRNPC1RAB9ANOTUMPTGS2
SCHEMBL28357214 0.80 ALDH1A1 (0.35) NPC1RAB9AMAPTMEN1GAA
SCHEMBL5797082 0.78 MAOB (0.35) NPC1RAB9AKDM4EMAPTPTGS2
SCHEMBL17047386 0.78 HSD17B10 (0.48) AHRCYP1B1NPC1RAB9ANOTUM
SCHEMBL10941967 0.78 AHR (0.46) AHRCYP1B1NPC1RAB9ANOTUM
SCHEMBL8529054 0.77 AHR (0.42) AHRCYP1B1NOTUMHTR2ASLC6A4
SCHEMBL9521923 0.77 NOTUM (0.35) NOTUMPTGS2KMO
SCHEMBL9649089 0.77 TSHR (0.32)
SCHEMBL7507597 0.76 GABRP (0.42) NPC1RAB9ANOTUMMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210179563-A1 PROCESS FOR THE MANUFACTURE OF IMINIUM COMPOUNDS AND THEIR APPLICATION IN THE MANUFACTURE OF PYRAZOLE DERIVATIVES SOLVAY SA (BE) 2021-06-17 US disclosed
US-20210171468-A1 PROCESS FOR THE MANUFACTURE OF PYRAZOLE CARBOXYLIC DERIVATIVES AND PRECURSORS THEREOF SOLVAY SA (BE) 2021-06-10 US disclosed
US-20200305431-A1 PROCESS FOR THE MANUFACTURE OF PYRAZOLE COMPOUNDS SOLVAY SA (BE) 2020-10-01 US disclosed
CN-111587242-A Process for producing pyrazole compound 索尔维公司 2020-08-25 CN disclosed
CN-111587241-A Method for producing iminium compound and use thereof for producing pyrazole derivative 索尔维公司 2020-08-25 CN disclosed
CN-111566093-A Method for producing pyrazolecarboxylic acid derivative and precursor thereof 索尔维公司 2020-08-21 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200305431-A1 PROCESS FOR THE MANUFACTURE OF PYRAZOLE COMPOUNDS CYP3A4, CYP3A43, CYP2E1 AHR 78/4885CYP1B1 9/4885NPC1 2185/4885
US-20210171468-A1 PROCESS FOR THE MANUFACTURE OF PYRAZOLE CARBOXYLIC DERIVATIVES AND PRECURSORS THEREOF CYP3A4, CYP3A43, CYP3A5 AHR 144/4885CYP1B1 15/4885NPC1 3582/4885
US-20210179563-A1 PROCESS FOR THE MANUFACTURE OF IMINIUM COMPOUNDS AND THEIR APPLICATION IN THE MANUFACTURE OF PYRAZOLE DERIVATIVES CYP3A5, CYP3A4, CYP3A43 AHR 481/4885CYP1B1 20/4885NPC1 3719/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.