SCHEMBL2246705

SCHEMBL2246705

C#Cc1ccc(-c2ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.60
CA1 P00915 4/20 0.60
ALB P02768 1/20 0.50
MMP2 P08253 2/20 0.46
MMP9 P14780 2/20 0.46
C3AR1 Q16581 1/20 0.45
KMT2A Q03164 1/20 0.44
MMP12 P39900 1/20 0.44
FOLH1 Q04609 2/20 0.43
FPGS Q05932 1/20 0.42
ADAMTS4 O75173 1/20 0.41
ADAMTS5 Q9UNA0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2246061 0.87 CA2 (0.69) CA2CA1MMP2MMP9C3AR1
SCHEMBL2245325 0.87 CA2 (0.69) CA2CA1MMP2MMP9C3AR1
SCHEMBL5508045 0.85 CA2 (0.61) CA2CA1ALBFOLH1
SCHEMBL2246702 0.85 MMP12 (0.60) CA2CA1ALBMMP2MMP12
SCHEMBL2245609 0.84 CA2 (0.66) CA2CA1MMP2MMP9C3AR1
SCHEMBL2249747 0.82 CA2 (0.63) CA2CA1MMP2MMP9C3AR1
SCHEMBL4621821 0.82 CA2 (0.63) CA2CA1MMP2MMP9C3AR1
SCHEMBL2242569 0.82 CA2 (0.63) CA2CA1C3AR1KMT2A
SCHEMBL2249692 0.81 CA2 (0.62) CA2CA1MMP2MMP9C3AR1
SCHEMBL2246916 0.81 CA2 (0.58) CA2CA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed