SCHEMBL2249692

SCHEMBL2249692

CCc1ccc(-c2ccc(C(=O)N[C@@H](CCC(N)=O)C(=O)O)cc2)cc1

nearest known ligand 0.62

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 9/20 0.62
CA1 P00915 5/20 0.62
TAS1R3 Q7RTX0 1/20 0.51
TAS1R1 Q7RTX1 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
MMP2 P08253 2/20 0.47
MMP9 P14780 2/20 0.47
CA12 O43570 1/20 0.46
CA9 Q16790 1/20 0.46
C3AR1 Q16581 1/20 0.46
DHFR P00374 2/20 0.46
TAOK1 Q7L7X3 1/20 0.46
TAOK3 Q9H2K8 1/20 0.46
TYMS P04818 1/20 0.46
KMT2A Q03164 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4621821 0.88 CA2 (0.63) CA2CA1MMP2MMP9C3AR1
SCHEMBL2246061 0.88 CA2 (0.69) CA2CA1NPC1RAB9AMMP2
SCHEMBL2245325 0.88 CA2 (0.69) CA2CA1NPC1RAB9AMMP2
SCHEMBL1096615 0.88 TAS1R3 (0.49) CA2CA1TAS1R3TAS1R1L3MBTL1
SCHEMBL4239668 0.86 TAS1R3 (0.50) CA2CA1TAS1R3TAS1R1L3MBTL1
SCHEMBL2245609 0.85 CA2 (0.66) CA2CA1MMP2MMP9C3AR1
SCHEMBL2249688 0.85 MMP12 (0.61) CA2CA1TAS1R3TAS1R1L3MBTL1
SCHEMBL2246916 0.84 CA2 (0.58) CA2CA1TAS1R3TAS1R1RAB9A
SCHEMBL2246508 0.84 CA2 (0.60) CA2CA1L3MBTL1NPC1RAB9A
SCHEMBL2249747 0.83 CA2 (0.63) CA2CA1MMP2MMP9C3AR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998965-B2 Glutamate aggrecanase inhibitors WYETH LLC (US) 2011-08-16 US disclosed