SCHEMBL22476545

SCHEMBL22476545

COC(C(C)C(C=O)Cc1ccccc1)C1CCCN1C=O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PREP P48147 1/20 0.36
CHRNB4 P30926 2/20 0.34
CHRNA3 P32297 2/20 0.34
MTNR1B P49286 1/20 0.33
GAA P10253 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
TAAR1 Q96RJ0 1/20 0.32
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22476487 0.89 PREP (0.37) PREPCHRNB4CHRNA3MTNR1BGAA
SCHEMBL18683750 0.78 NPC1 (0.41) PREPGAAMEN1KMT2ATAAR1
SCHEMBL22476440 0.77 F2 (0.38) PREPGAAMEN1KMT2AATM
SCHEMBL23154537 0.77 ACE (0.46) GAAKMT2AMAPK1ACE
SCHEMBL25949990 0.77 ACE (0.46) GAAKMT2AMAPK1ACE
SCHEMBL18688556 0.77 ACE (0.46) GAAKMT2AMAPK1ACE
SCHEMBL21699258 0.76 CYP2C9 (0.49) GAAATML3MBTL1TSHR
SCHEMBL21699268 0.76 CYP2C9 (0.49) GAAATML3MBTL1TSHR
SCHEMBL21335916 0.76 PREP (0.46) PREPTSHRACE
SCHEMBL22476544 0.75 MMP1 (0.44) ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3303366-B1 DERIVATIVES OF DOLASTATIN 10 AND USES THEREOF NEWBIO THERAPEUTICS INC (CN) 2020-09-30 EP disclosed