SCHEMBL22482913

SCHEMBL22482913

NC(=O)c1ccc(CN(Sc2cc(F)c(F)c(F)c2F)C2CC2)cc1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 15/20 0.43
HDAC8 Q9BY41 11/20 0.43
HDAC11 Q96DB2 4/20 0.38
HDAC3 O15379 3/20 0.38
KCNA5 P22460 1/20 0.35
NSD2 O96028 1/20 0.34
HDAC2 Q92769 1/20 0.34
DPP4 P27487 1/20 0.33
DPP8 Q6V1X1 1/20 0.33
DPP9 Q86TI2 1/20 0.33
DPP7 Q9UHL4 1/20 0.33
DRD3 P35462 1/20 0.33
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24472873 0.86 HDAC6 (0.60) HDAC6HDAC8HDAC11HDAC3HDAC2
SCHEMBL20847480 0.84 HDAC6 (0.43) HDAC6HDAC8HDAC11HDAC3KCNA5
SCHEMBL24473206 0.82 HDAC6 (0.48) HDAC6HDAC8HDAC11HDAC3HDAC2
SCHEMBL24472776 0.78 HDAC6 (0.59) HDAC6HDAC8HDAC11HDAC3HDAC2
SCHEMBL22482914 0.76 HDAC6 (0.37) HDAC6HDAC8HDAC3HDAC2
SCHEMBL24473211 0.75 HDAC6 (0.54) HDAC6HDAC8HDAC11HDAC3HDAC2
SCHEMBL20847775 0.73 KMT2A (0.44) HDAC6HDAC8HDAC11HDAC3NSD2
SCHEMBL20847600 0.71 HDAC8 (0.43) HDAC6HDAC8HDAC11HDAC3
SCHEMBL24473070 0.70 HDAC6 (0.61) HDAC6HDAC8HDAC11HDAC3
SCHEMBL20847479 0.68 HDAC6 (0.74) HDAC6HDAC8HDAC11HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020194272-A1 HALOGENATED PHENYLSULFONAMIDE HYDROXAMIC ACID COMPOUNDS, COMPOSITIONS AND USES THEREOF AS SELECTIVE HDAC6 INHIBITORS 2681603 ONTARIO INC. (CA) 2020-10-01 WO disclosed