SCHEMBL22487927

SCHEMBL22487927

CC(C)c1nc2c(=O)n(-c3ccncc3)cnc2[nH]1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.41
KDM5B Q9UGL1 2/20 0.36
GRM1 Q13255 4/20 0.34
GRM5 P41594 1/20 0.33
XDH P47989 3/20 0.32
CYP17A1 P05093 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CNOT7 Q9UIV1 1/20 0.31
HCAR1 Q9BXC0 1/20 0.30
PDE2A O00408 1/20 0.30
MCHR1 Q99705 1/20 0.30
AR P10275 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22487919 0.79 GRM1 (0.35) GRM1GRM5XDHCYP17A1NPSR1
SCHEMBL5432319 0.68 GRM1 (0.42) GRM1GRM5PDE2A
SCHEMBL22487747 0.67 XDH (0.42) GRM1XDHHCAR1
SCHEMBL5437218 0.66 MEN1 (0.46) GRM1GRM5XDHHCAR1
SCHEMBL24422535 0.64 GSK3B (0.36) GSK3B
SCHEMBL22488037 0.63 HPGD (0.39) GRM1XDHHCAR1
SCHEMBL22487730 0.63 ACHE (0.37) GSK3BXDHNPSR1
SCHEMBL3992299 0.62 GSK3B (0.32) GSK3B
SCHEMBL11003505 0.60 GSK3B (0.43) GSK3B
SCHEMBL10537854 0.59 MAT2A (0.33) GRM1CYP17A1AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20200308165-A1 Compounds as Ras Inhibitors and Use Thereof D. E. SHAW RESEARCH, LLC 2020-10-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200308165-A1 Compounds as Ras Inhibitors and Use Thereof KRAS, NRAS, HRAS GSK3B 2312/4885KDM5B 4047/4885GRM1 4660/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.