SCHEMBL224929

SCHEMBL224929

CC(C)(C)OC(=O)NC1CCC(CC=O)CC1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.51
DRD2 P14416 8/20 0.47
BTK Q06187 1/20 0.47
KDM1A O60341 1/20 0.44
MAOB P27338 1/20 0.44
CTSK P43235 2/20 0.43
DRD3 P35462 2/20 0.43
GAA P10253 2/20 0.42
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
KMT2A Q03164 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11921121 1.00 EPHX1 (0.51) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL224930 1.00 EPHX1 (0.51) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL2977422 0.86 DRD2 (0.48) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL2977423 0.86 DRD2 (0.48) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL34465370 0.86 BTK (0.48) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL15662556 0.86 BTK (0.48) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL8074670 0.85 EPHX1 (0.46) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL28984107 0.85 EPHX1 (0.46) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL20051778 0.85 EPHX1 (0.46) EPHX1DRD2BTKKDM1AMAOB
SCHEMBL28984106 0.85 EPHX1 (0.46) EPHX1DRD2BTKKDM1AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 194 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260109708-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS DEGRADERS OF MK2 KINASE CELGENE CORP (US) 2026-04-23 US disclosed
EP-4662207-A2 COMPOUNDS AND COMPOSITIONS USEFUL AS DEGRADERS OF MK2 KINASE Celgene Corporation (US) 2025-12-17 EP disclosed
WO-2025230799-A2 CYCLOALKYL- AND PIPERIDINYL-CONTAINING DIAMINOMETHYLENE PYRIMIDINE-2,4,6-TRIONE AGONISTS OF PARATHYROID HORMONE 1 AND INCRETIN RECEPTORS SEPTERNA, INC. (US) 2025-11-06 WO disclosed
US-20250326729-A1 PROCESS FOR THE PREPARATION OF CARIPRAZINE F.I.S. FABBRICA ITALIANA SINTETICI S.P.A. (IT) 2025-10-23 US disclosed
US-20250326764-A1 INHIBITORS OF THE MENIN-MLL INTERACTION VITAE PHARMACEUTICALS LLC (US) 2025-10-23 US disclosed
EP-4635946-A1 IMPROVED PROCESS FOR THE PREPARATION OF CARIPRAZINE F.I.S. Fabbrica Italiana Sintetici S.p.A. (IT) 2025-10-22 EP disclosed
EP-4608810-A1 COMPOUNDS, COMPOSITIONS AND METHODS OF USE TO TREAT HYPOPARATHYROIDISM AND OSTEOPOROSIS Septerna, Inc. (US) 2025-09-03 EP disclosed
WO-2025129168-A1 TRIAZOLONE INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE AND THEIR THERAPEUTIC USES THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2025-06-19 WO disclosed
EP-4558495-A1 HETEROARYL COMPOUNDS AS LIGAND DIRECTED DEGRADERS OF IRAK4 Bristol-Myers Squibb Company (US) 2025-05-28 EP disclosed
US-12312359-B2 Inhibitors of the menin-MLL interaction VITAE PHARMACEUTICALS, LLC (US) 2025-05-27 US disclosed
EP-1725238-A2 M 3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2006-11-29 EP disclosed
EP-1725564-A1 M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2006-11-29 EP disclosed
US-20060211758-A1 M3 muscarinic acetylcholine receptor antagonists SMITHKLINE BEECHAM CORPORATION 2006-09-21 US disclosed
EP-1613307-A2 M SB 3 /SB MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2006-01-11 EP disclosed
WO-2005094251-A2 M3MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2005-10-13 WO disclosed
WO-2005095407-A1 M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2005-10-13 WO disclosed
WO-2004091482-A2 M3 MUSCARINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS GLAXO GROUP LIMITED (GB) 2004-10-28 WO disclosed
CN-1329609-A Tetrahydrobenza epine derivatives useful as modulators of dopamine D3 receptors (antipsychotic agents) SMITHKLINE BEECHAM PLC (GB) 2002-01-02 CN disclosed
EP-0983244-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS SMITHKLINE BEECHAM PLC (GB) 2000-03-08 EP disclosed
WO-1998050364-A1 TETRAHYDROISOQUINOLINE DERIVATIVES AS MODULATORS OF DOPAMINE D3 RECEPTORS SMITHKLINE BEECHAM PLC (GB) 1998-11-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060211758-A1 M3 muscarinic acetylcholine receptor antagonists CHRM3, CHRM2, CHRM5 EPHX1 2067/4885DRD2 859/4885BTK 3429/4885
US-12312359-B2 Inhibitors of the menin-MLL interaction MLLT1, MEN1, MLLT3 EPHX1 2775/4885DRD2 4732/4885BTK 2479/4885
US-20250326729-A1 PROCESS FOR THE PREPARATION OF CARIPRAZINE CYP3A5, CYP4Z1, FIP1L1 EPHX1 832/4885DRD2 821/4885BTK 4527/4885
US-20260109708-A1 COMPOUNDS AND COMPOSITIONS USEFUL AS DEGRADERS OF MK2 KINASE PSME2, MKRN3, RPS6KA2 EPHX1 3853/4885DRD2 3260/4885BTK 1312/4885
US-20250326764-A1 INHIBITORS OF THE MENIN-MLL INTERACTION MLLT1, MEN1, MLLT3 EPHX1 2775/4885DRD2 4732/4885BTK 2479/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.