SCHEMBL22506486

SCHEMBL22506486

COC(=O)c1ccc(/C=N/c2c(N)[nH]c(=S)[nH]c2=O)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIG1 P18858 1/20 0.63
LIG3 P49916 1/20 0.63
LIG4 P49917 1/20 0.63
CA1 P00915 3/20 0.48
CA2 P00918 3/20 0.48
PTGS2 P35354 2/20 0.46
PTGS1 P23219 1/20 0.46
G6PD P11413 1/20 0.46
GRIN2D O15399 1/20 0.45
GRIN3B O60391 1/20 0.45
GRIN1 Q05586 1/20 0.45
GRIN2A Q12879 1/20 0.45
GRIN2B Q13224 1/20 0.45
GRIN2C Q14957 1/20 0.45
GRIN3A Q8TCU5 1/20 0.45
TDP1 Q9NUW8 1/20 0.42
KDM4E B2RXH2 3/20 0.42
RXFP1 Q9HBX9 1/20 0.42
MAPT P10636 2/20 0.41
ALDH1A1 P00352 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22506412 0.83 LIG1 (0.69) LIG1LIG3LIG4CA2PTGS2
SCHEMBL13934092 0.70 CA2 (0.88) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11409395 0.70 CA1 (0.62) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11409392 0.70 CA1 (0.62) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11418984 0.69 CA1 (0.58) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11411393 0.69 CA1 (0.65) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11422967 0.69 CA1 (0.61) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11411395 0.69 CA1 (0.65) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11418985 0.69 CA1 (0.58) CA1CA2PTGS2PTGS1GRIN2D
SCHEMBL11415365 0.68 CA1 (0.56) CA1CA2PTGS2PTGS1GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220162649-A1 NOVEL NUCLEIC ACID MODIFIERS NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-05-26 US disclosed
WO-2020206036-A1 NOVEL NUCLEIC ACID MODIFIER THE BROAD INSTITUTE, INC. (US) 2020-10-08 WO disclosed