SCHEMBL225527

SCHEMBL225527

FC(F)(F)c1[c]cccc1Cl

nearest known ligand 0.33

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.33
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3583635 0.82 CYP2A6 (0.38) TSHRLMNA
SCHEMBL979836 0.81 PDK2 (0.39)
SCHEMBL15638416 0.78 GPBAR1 (0.36)
SCHEMBL3109144 0.77 LMNA (0.33) TSHRLMNA
SCHEMBL5314612 0.74 CYP3A4 (0.41) TSHR
SCHEMBL81364 0.74
SCHEMBL82438 0.74 TDP1 (0.34) LMNA
SCHEMBL15636512 0.74 GPBAR1 (0.39)
SCHEMBL15637459 0.73 HSD11B1 (0.42) TSHR
SCHEMBL6591152 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 629 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024102177-A1 COMBINATION THERAPIES FOR THE TREATMENT OF BRAIN CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-05-16 WO claimed
WO-2024081447-A1 EGFR INHIBITORS FOR TREATING LUNG CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2024-04-18 WO claimed
EP-4345101-A1 AZOLE DERIVATIVES AS SHP2 INHIBITORS IRBM S.P.A. (IT) 2024-04-03 EP claimed
WO-2023244639-A1 METHODS OF PREDICTING CNS CANCER RESPONSE TO TREATMENT WITH EGFR INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2023-12-21 WO claimed
WO-2023239768-A1 TRICYCLIC TRIAZOLO COMPOUNDS AS DGK INHIBITORS INCYTE CORPORATION (US) 2023-12-14 WO claimed
US-20230399342-A1 TRICYCLIC TRIAZOLO COMPOUNDS AS DGK INHIBITORS INCYTE CORPORATION 2023-12-14 US claimed
US-20230364091-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER THE REGENTS OF THE UNIVERSITY OF CALIFORNIA 2023-11-16 US claimed
EP-3867238-B1 PROTEIN TYROSINE PHOSPHATASE INHIBITORS ARRAY BIOPHARMA INC (US) 2023-06-07 EP claimed
CN-114341124-A Protein tyrosine phosphatase inhibitors ARRAY生物制药公司 2022-04-12 CN claimed
CN-113811528-A Compositions and methods for treating cancer 加利福尼亚大学董事会 2021-12-17 CN claimed
US-4582906-A REDUCED SOIL BIODEGRADATION OF THIOL CARBAMATES STAUFFER CHEMICAL COMPANY (US) 1986-04-15 US claimed
US-4542126-A Pesticidally active pyrimidin-5-yl-(thio)phosphoric acid ester-amides BAYER AKTIENGESELLSCHAFT (DE) 1985-09-17 US claimed
US-4540429-A 4-Phenyl-1,2,3-thiadiazoles as herbicide extenders STAUFFER CHEMICAL COMPANY (US) 1985-09-10 US claimed
US-4512989-A IMIDOESTERS OR IMIDOTHIOESTERS HOKKO CHEMICAL INDUSTRY CO., LTD. (JP) 1985-04-23 US claimed
EP-0062773-B1 4-Phenyl-1,2,3-thiadiazoles as herbicide extenders STAUFFER CHEMICAL COMPANY (US) 1984-12-05 EP claimed
EP-0118864-A1 Pyrimidinyl derivatives BAYER AG (DE) 1984-09-19 EP claimed
US-4391804-A Imidazole derivatives and fungicidal composition containing the same HOKKO CHEMICAL INDUSTRY COMPANY, LTD. (JP) 1983-07-05 US claimed
EP-0062773-A1 4-Phenyl-1,2,3-thiadiazoles as herbicide extenders STAUFFER CHEMICAL COMPANY (US) 1982-10-20 EP claimed
US-4146386-A Phthalic dianilides and their use as plant growth regulators MONSANTO COMPANY (US) 1979-03-27 US claimed
US-4016281-A Tetralone and indanone compounds MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DT) 1977-04-05 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230364091-A1 COMPOSITIONS AND METHODS FOR TREATING CANCER TP53, EGFR, SLC2A1 TSHR 3410/4885LMNA 3720/4885
US-20230399342-A1 TRICYCLIC TRIAZOLO COMPOUNDS AS DGK INHIBITORS DGKA, DGKI, DGKG TSHR 2904/4885LMNA 2825/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.