SCHEMBL22554085

SCHEMBL22554085

Cn1cc(C(=O)O)c2c(Cl)ccnc21

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 4/20 0.40
KDM4E B2RXH2 3/20 0.40
KDM5A P29375 2/20 0.40
KDM6B O15054 1/20 0.40
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
CYP2C9 P11712 2/20 0.37
MEN1 O00255 1/20 0.37
POLB P06746 1/20 0.37
KMT2A Q03164 1/20 0.37
FTO Q9C0B1 2/20 0.36
SORT1 Q99523 3/20 0.36
DHODH Q02127 1/20 0.35
ALDH1A1 P00352 2/20 0.35
CAMKK1 Q8N5S9 1/20 0.34
CAMKK2 Q96RR4 1/20 0.34
KDM2B Q8NHM5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26457800 0.88 KDM4E (0.42) KDM4CKDM4EKDM5AKDM6BLMNA
SCHEMBL31277771 0.81 KDM5A (0.38) KDM4CKDM4EKDM5ALMNASMN1; SMN2
SCHEMBL17818874 0.78 CNR1 (0.47) KDM4C
SCHEMBL3690474 0.78 LMNA (0.41) KDM4CKDM4EKDM5ALMNASMN1; SMN2
SCHEMBL23910951 0.76 L3MBTL1 (0.43) KDM4EPTGDR2POLBALDH1A1
SCHEMBL1229639 0.76 SRC (0.36) KDM4CKDM4EKDM5AKDM6BLMNA
SCHEMBL17818705 0.76 KDM4E (0.34) KDM4CKDM4EKDM5ALMNASMN1; SMN2
SCHEMBL22729832 0.75 LMNA (0.45) KDM4CKDM4EKDM5ALMNASMN1; SMN2
SCHEMBL29912799 0.75 LMNA (0.45) KDM4CKDM4EKDM5ALMNASMN1; SMN2
SCHEMBL17518149 0.75 CDK5 (0.35) PTGDR2POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11919902-B2 Aryl-bipyridine amine derivatives as phosphatidylinositol phosphate kinase inhibitors HIBERCELL, INC. (US) 2024-03-05 US disclosed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed
CN-112088157-A Aryl-bipyridine amine derivatives as phosphoinositide kinase inhibitors 拉文纳制药公司 2020-12-15 CN disclosed
US-20200331913-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS HIBERCELL, INC. 2020-10-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200331913-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS PIP5K1A, PIP5K1B, PIP5K1C KDM4C 1727/4885KDM4E 774/4885KDM5A 819/4885
US-11919902-B2 Aryl-bipyridine amine derivatives as phosphatidylinositol phosphate kinase inhibitors PIP5K1A, PIP5K1B, PIP5K1C KDM4C 1727/4885KDM4E 774/4885KDM5A 819/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.