SCHEMBL22554150

SCHEMBL22554150

O=C1CCCN1c1ccc(-c2cncc(-c3cn(Cc4ccccc4)c(=O)c4[nH]ncc34)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 1/20 0.40
BRD4 O60885 1/20 0.39
BRDT Q58F21 1/20 0.39
CCNC P24863 1/20 0.39
CDK8 P49336 1/20 0.39
P2RX7 Q99572 1/20 0.38
CDK2 P24941 2/20 0.38
PARP1 P09874 1/20 0.37
PRKAB2 O43741 1/20 0.36
PRKAG1 P54619 1/20 0.36
PRKAA2 P54646 1/20 0.36
PRKAA1 Q13131 1/20 0.36
PRKAG3 Q9UGI9 1/20 0.36
PRKAG2 Q9UGJ0 1/20 0.36
PRKAB1 Q9Y478 1/20 0.36
USP1 O94782 1/20 0.36
FNTA P49354 1/20 0.35
PGGT1B P53609 1/20 0.35
CYP11B1 P15538 1/20 0.35
CYP11B2 P19099 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22554295 0.86 BRD4 (0.48) BRD4BRDTCCNCCDK8PRKAB2
SCHEMBL22554262 0.85 CCNC (0.39) BRD4BRDTCCNCCDK8CDK2
SCHEMBL22554090 0.82 METAP2 (0.37) CDC7BRD4BRDTCCNCCDK8
SCHEMBL22554254 0.77 PRKAB2 (0.41) CCNCCDK8PARP1PRKAB2PRKAG1
SCHEMBL28563220 0.75 CYP11B1 (0.42) CDC7CCNCCDK8P2RX7CDK2
SCHEMBL22553792 0.74 SMN1; SMN2 (0.41) CCNCCDK8CYP11B1CYP11B2NPC1
SCHEMBL30730803 0.74 SMN1; SMN2 (0.41) CCNCCDK8CYP11B1CYP11B2NPC1
SCHEMBL22553760 0.73 PRKAB2 (0.40) CCNCCDK8PRKAB2PRKAG1PRKAA2
SCHEMBL30730822 0.73 PRKAB2 (0.40) CCNCCDK8PRKAB2PRKAG1PRKAA2
SCHEMBL22553955 0.72 PIM1 (0.42) BRD4CCNCCDK8CYP11B2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN claimed
EP-3728230-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS Ravenna Pharmaceuticals, Inc. (US) 2020-10-28 EP claimed
US-20200331913-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS HIBERCELL, INC. 2020-10-22 US claimed
US-11919902-B2 Aryl-bipyridine amine derivatives as phosphatidylinositol phosphate kinase inhibitors HIBERCELL, INC. (US) 2024-03-05 US disclosed
CN-112088157-B Aryl-bipyridylamine derivatives as phosphatidylinositol phosphokinase inhibitors 拉文纳制药公司 2023-12-26 CN disclosed
EP-3728230-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS Ravenna Pharmaceuticals, Inc. (US) 2020-10-28 EP disclosed
US-20200331913-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS HIBERCELL, INC. 2020-10-22 US disclosed
US-20200331913-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS HIBERCELL, INC. 2020-10-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20200331913-A1 ARYL-BIPYRIDINE AMINE DERIVATIVES AS PHOSPHATIDYLINOSITOL PHOSPHATE KINASE INHIBITORS PIP5K1A, PIP5K1B, PIP5K1C CDC7 681/4885BRD4 309/4885BRDT 786/4885
US-11919902-B2 Aryl-bipyridine amine derivatives as phosphatidylinositol phosphate kinase inhibitors PIP5K1A, PIP5K1B, PIP5K1C CDC7 681/4885BRD4 309/4885BRDT 786/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.