SCHEMBL22558366

SCHEMBL22558366

CCOC(=O)C(N=C(c1ccccc1)c1ccccc1)c1cnc(Cl)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
NPC1 O15118 2/20 0.43
DGAT1 O75907 1/20 0.37
TBXAS1 P24557 2/20 0.37
SMN1; SMN2 Q16637 4/20 0.36
RAB9A P51151 2/20 0.36
GAA P10253 1/20 0.36
AAK1 Q2M2I8 1/20 0.36
PIN1 Q13526 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
ALDH1A1 P00352 3/20 0.35
MAPT P10636 2/20 0.35
LMNA P02545 1/20 0.34
MAPK1 P28482 1/20 0.34
ATM Q13315 1/20 0.34
POLB P06746 1/20 0.34
PKM P14618 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29473304 1.00 MEN1 (0.43) MEN1KMT2ANPC1DGAT1TBXAS1
SCHEMBL26670573 0.86 MEN1 (0.43) MEN1KMT2ANPC1TBXAS1SMN1; SMN2
SCHEMBL4469552 0.82 TBXAS1 (0.45) MEN1KMT2ANPC1TBXAS1SMN1; SMN2
SCHEMBL26693677 0.82 KMT2A (0.41) MEN1KMT2ANPC1TBXAS1SMN1; SMN2
SCHEMBL28698607 0.78 AAK1 (0.35) TBXAS1AAK1ALDH1A1MAPTLMNA
SCHEMBL26693982 0.76 MEN1 (0.42) MEN1KMT2ANPC1TBXAS1SMN1; SMN2
SCHEMBL17018473 0.75 KMT2A (0.43) MEN1KMT2ANPC1TBXAS1AAK1
SCHEMBL26670483 0.75 TSHR (0.44) MEN1KMT2ANPC1TBXAS1SMN1; SMN2
SCHEMBL29837799 0.74 KMT2A (0.40) MEN1KMT2ANPC1TBXAS1SMN1; SMN2
SCHEMBL26693646 0.74 KMT2A (0.40) MEN1KMT2ANPC1TBXAS1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4526298-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS F. Hoffmann-La Roche AG (CH) 2025-03-26 EP disclosed
US-20250074913-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS HOFFMANN-LA ROCHE INC. (US) 2025-03-06 US disclosed
US-11845752-B2 Substituted imidazo[1,5-a]pyrazines for the treatment of hepatitis B ALIGOS THERAPEUTICS, INC. (US) 2023-12-19 US disclosed
WO-2023222644-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2023-11-23 WO disclosed
WO-2023222644-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2023-11-23 WO disclosed
EP-4229062-A1 BICYCLIC COMPOUNDS Aligos Therapeutics, Inc. (US) 2023-08-23 EP disclosed
US-11591341-B2 Bicyclic and tricyclic compounds ALIGOS THERAPEUTICS, INC. (US) 2023-02-28 US disclosed
US-20220119395-A1 BICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2022-04-21 US disclosed
WO-2022081758-A1 BICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. (US) 2022-04-21 WO disclosed
EP-3956331-A1 BICYCLIC AND TRICYCLIC COMPOUNDS Aligos Therapeutics, Inc. (US) 2022-02-23 EP disclosed
US-20200361947-A1 BICYCLIC AND TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. 2020-11-19 US disclosed
WO-2020214728-A1 BICYCLIC AND TRICYCLIC COMPOUNDS ALIGOS THERAPEUTICS, INC. (US) 2020-10-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11845752-B2 Substituted imidazo[1,5-a]pyrazines for the treatment of hepatitis B SLC10A1, HAVCR2, CYP3A5 MEN1 2681/4885KMT2A 3209/4885NPC1 69/4885
US-20220119395-A1 BICYCLIC COMPOUNDS SLC10A1, PKD1, CYP11B2 MEN1 262/4885KMT2A 3870/4885NPC1 11/4885
US-20200361947-A1 BICYCLIC AND TRICYCLIC COMPOUNDS SLC10A1, PKD1, CYP11B2 MEN1 376/4885KMT2A 3587/4885NPC1 15/4885
US-20250074913-A1 PYRAZOLE DERIVATIVES AS STING AGONISTS STING1, CGAS, MAVS MEN1 2237/4885KMT2A 4029/4885NPC1 1915/4885
US-11591341-B2 Bicyclic and tricyclic compounds SLC10A1, PKD1, CYP11B2 MEN1 376/4885KMT2A 3587/4885NPC1 15/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.