Imidazole

Imidazole

SCHEMBL2256134

CC(=O)O.Cl.c1c[nH]cn1

nearest known ligand 0.62

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Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Imidazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.62
FKBP5 Q13451 1/20 0.62
FFAR3 O14843 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Imidazole SCHEMBL145932 0.98
Imidazole SCHEMBL29411697 0.98 ALDH1A1 (0.65) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL28966030 0.98 ALDH1A1 (0.65) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL30320112 0.98 ALDH1A1 (0.65) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL3639063 0.95 ALDH1A1 (0.62) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL29365438 0.95 ALDH1A1 (0.62) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL29188028 0.95 ALDH1A1 (0.62) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL28796723 0.95 ALDH1A1 (0.62) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL27735299 0.95 ALDH1A1 (0.62) ALDH1A1FKBP5FFAR3LCKFYN
Imidazole SCHEMBL28213689 0.95 ALDH1A1 (0.62) ALDH1A1FKBP5FFAR3LCKFYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112574113-A Zoledronic acid intermediate compound 鲁南制药集团股份有限公司 2021-03-30 CN disclosed
CN-102553645-B Ionic liquid 2-(1-imidazolyl)-supported acetate catalyst and preparation method thereof NANJING UNIVERSITY OF TECHNOLOGY 2013-10-09 CN disclosed
CN-102775444-A New preparation method of zoledronic acid HENGSHUI KANGYI MEDICAL TECHNOLOGY DEV CO LTD 2012-11-14 CN disclosed
CN-102553645-A Ionic liquid 2-(1-imidazolyl)-supported acetate catalyst and preparation method thereof NANJING UNIVERSITY OF TECHNOLOGY 2012-07-11 CN disclosed
US-20110206617-A1 MODIFIED POLYSACCHARIDES FOR DRUG AND CONTRAST AGENT DELIVERY WILLIAM MARSH RICE UNIVERSITY 2011-08-25 US disclosed
CN-101223143-A 3-cyanoquinoline inhibitors of TPL2 kinase and methods of making and using the same WYETH CORP (US) 2008-07-16 CN disclosed
CN-1693308-A Process for preparing dazoline phospho acid YANGZIJIANG PHARMACEUTICAL GRO (CN) 2005-11-09 CN disclosed
CN-1472215-A Synthesis of product prepared from imidazole acted with halogenated acetate ethyl ester 武汉麦林新技术开发有限公司 2004-02-04 CN disclosed
EP-0618913-B1 IMIDAZOLYL OR IMIDAZOYLALKYL SUBSTITUTED WITH A FOUR OR FIVE MEMBERED NITROGEN CONTAINING HETEROCYCLIC RING SCHERING CORP (US) 1996-08-14 EP disclosed
US-5463074-A Treating allergy, inflammation, hypertension, glaucoma, central nervous system disorders SCHERING CORPORATION (US) 1995-10-31 US disclosed
EP-0533242-A2 Substituted derivatives of piperazinylcamphorsulfonyl oxytocin antagonists MERCK & CO. INC. (US) 1993-03-24 EP disclosed