SCHEMBL22562432

SCHEMBL22562432

N#Cc1cc(-n2c3ccccc3c3ccc(-c4ccccc4C#N)cc32)c(-c2cccc(-c3ccccc3)n2)c(-n2c3ccccc3c3ccc(-c4ccccc4C#N)cc32)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRG2 P18507 7/20 0.38
GABRB3 P28472 7/20 0.38
GABRA5 P31644 5/20 0.38
GABRA3 P34903 5/20 0.38
TRPA1 O75762 1/20 0.37
GABRA1 P14867 6/20 0.36
GABRA2 P47869 4/20 0.36
NR3C1 P04150 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
CYP19A1 P11511 1/20 0.34
CYP1A2 P05177 3/20 0.33
CYP3A4 P08684 3/20 0.33
LMNA P02545 2/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562431 0.95 GABRG2 (0.35) GABRG2GABRB3GABRA5GABRA3TRPA1
SCHEMBL22562267 0.92 ALDH1A3 (0.34) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL22562451 0.91 GABRG2 (0.40) GABRG2GABRB3GABRA5GABRA3TRPA1
SCHEMBL22562272 0.89 ALDH1A3 (0.36) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL22562396 0.89 GABRG2 (0.38) GABRG2GABRB3GABRA5GABRA3TRPA1
SCHEMBL22562448 0.88 ALDH1A3 (0.45) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL22562258 0.88 ALDH1A3 (0.40) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL22562282 0.87 PTGER4 (0.35) GABRG2GABRB3GABRA5GABRA3GABRA1
SCHEMBL19919474 0.85 GABRG2 (0.41) GABRG2GABRB3GABRA5GABRA3TRPA1
SCHEMBL21546720 0.85 ADRA2C (0.37) GABRG2GABRB3GABRA5GABRA3TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3418278-B1 ORGANIC MOLECULES, IN PARTICULAR FOR USE IN OPTOELECTRONIC DEVICES CYNORA GMBH (DE) 2020-10-21 EP disclosed