SCHEMBL22562939

SCHEMBL22562939

CC(=N)c1ccc(Nc2c(F)cccc2Cl)cc1N

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.38
ABCB11 O95342 1/20 0.38
PTGS1 P23219 1/20 0.38
PPARG P37231 1/20 0.38
NR1I3 Q14994 1/20 0.38
HDAC1 Q13547 1/20 0.37
RAPGEF4 Q8WZA2 2/20 0.36
CHRNA7 P36544 6/20 0.36
JAK1 P23458 2/20 0.35
JAK3 P52333 2/20 0.35
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
FADS1 O60427 1/20 0.34
JAK2 O60674 1/20 0.34
TYK2 P29597 1/20 0.34
MAPK14 Q16539 2/20 0.34
MAPK13 O15264 1/20 0.34
MAPK12 P53778 1/20 0.34
MAPK11 Q15759 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562988 0.79 MAPK14 (0.47) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL22563179 0.79 HDAC1 (0.44) HDAC1MAPK14MAPK13MAPK12MAPK11
SCHEMBL22563163 0.75 HDAC1 (0.40) HDAC1
SCHEMBL22563042 0.75 PYGL (0.44) HDAC1TDO2MAPK14MAPK13MAPK12
SCHEMBL22563010 0.72 HDAC6 (0.37) HDAC1RAPGEF4CHRNA7JAK1JAK3
SCHEMBL22563002 0.71 MAP2K2 (0.41) HDAC1IDO1MAPK14MAPK13MAPK12
SCHEMBL22563186 0.71 JAK1 (0.37) HDAC1CHRNA7JAK1JAK3JAK2
SCHEMBL22562958 0.71 JAK1 (0.37) HDAC1JAK1JAK3JAK2TYK2
SCHEMBL1033031 0.70 PTGS2 (0.50) PTGS2ABCB11PTGS1PPARGNR1I3
Acetic Acid SCHEMBL28632464 0.69 PTGS2 (0.56) PTGS2ABCB11PTGS1PPARGNR1I3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed