SCHEMBL22563034

SCHEMBL22563034

CCCC(CCC)c1ccc(C(=O)NC(=N)c2ccc(Nc3c(F)cccc3CC)cc2N)cc1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 11/20 0.37
HDAC3 O15379 5/20 0.33
HDAC2 Q92769 5/20 0.33
NCOR2 Q9Y618 4/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
JAK2 O60674 2/20 0.32
JAK1 P23458 3/20 0.32
JAK3 P52333 3/20 0.32
TYK2 P29597 2/20 0.32
HDAC6 Q9UBN7 1/20 0.32
F2 P00734 1/20 0.30
F10 P00742 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22564663 0.96 HDAC1 (0.34) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22563017 0.92 HDAC1 (0.37) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22564672 0.92 HDAC1 (0.35) HDAC1JAK2JAK1JAK3TYK2
SCHEMBL22563185 0.78 HDAC1 (0.33) HDAC1HDAC3HDAC2KDM4EALDH1A1
SCHEMBL22563186 0.78 JAK1 (0.37) HDAC1KDM4EALDH1A1JAK2JAK1
SCHEMBL22562998 0.76 MAPK14 (0.33) HDAC1HDAC3HDAC2NCOR2
SCHEMBL22562958 0.76 JAK1 (0.37) HDAC1KDM4EALDH1A1JAK2JAK1
SCHEMBL22563056 0.72 HDAC1 (0.41) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22564671 0.69 HDAC8 (0.34) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22563010 0.66 HDAC6 (0.37) HDAC1JAK1JAK3TYK2HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed