SCHEMBL22563056

SCHEMBL22563056

CCCCC(CCC)c1ccc(C(=O)N/C(=C(/C)CC)c2ccc(Nc3cccc(F)c3)cc2N)cc1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.41
HDAC3 O15379 5/20 0.34
HDAC2 Q92769 5/20 0.34
NCOR2 Q9Y618 5/20 0.34
LMNA P02545 1/20 0.32
KMT2A Q03164 3/20 0.32
SNCA P37840 1/20 0.32
NPC1 O15118 3/20 0.32
RAB9A P51151 3/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 2/20 0.32
HPGD P15428 1/20 0.32
DGAT1 O75907 1/20 0.32
MAPT P10636 1/20 0.32
F2R P25116 1/20 0.32
PTGER4 P35408 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22562963 0.82 MAPK14 (0.39) HDAC1HDAC3HDAC2KMT2ANPC1
SCHEMBL22563017 0.72 HDAC1 (0.37) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22563034 0.72 HDAC1 (0.37) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22562998 0.71 MAPK14 (0.33) HDAC1HDAC3HDAC2NCOR2
SCHEMBL22564663 0.69 HDAC1 (0.34) HDAC1HDAC3HDAC2NCOR2KDM4E
SCHEMBL22563055 0.68 TBXA2R (0.38) HDAC1KMT2AMEN1MAPT
SCHEMBL22562973 0.67 MAPT (0.36) KMT2ANPC1KDM4EMEN1MAPT
SCHEMBL21732183 0.63 OPRM1 (0.42)
SCHEMBL28533240 0.61 BDKRB2 (0.49) LMNAHPGD
SCHEMBL22563037 0.60 RARB (0.47) KMT2AMEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed