SCHEMBL22562998

SCHEMBL22562998

CCCCCC(CCC)c1ccc(C(=O)NC(=N)c2ccc(Nc3ccccc3P)cc2N)cc1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 5/20 0.33
MAPK13 O15264 2/20 0.33
MAPK12 P53778 2/20 0.33
MAPK11 Q15759 2/20 0.33
HDAC1 Q13547 11/20 0.33
HDAC3 O15379 4/20 0.33
HDAC2 Q92769 4/20 0.33
PPARG P37231 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
ITGB3 P05106 1/20 0.31
ITGA2B P08514 1/20 0.31
NCOR2 Q9Y618 3/20 0.31
PLK1 P53350 2/20 0.30
PLK3 Q9H4B4 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22563043 0.86 ALDH1A1 (0.35) HDAC1HDAC3HDAC2PLK1PLK3
SCHEMBL22562963 0.80 MAPK14 (0.39) MAPK14MAPK13MAPK12MAPK11HDAC1
SCHEMBL22563017 0.77 HDAC1 (0.37) MAPK14MAPK13MAPK12MAPK11HDAC1
SCHEMBL22563034 0.76 HDAC1 (0.37) HDAC1HDAC3HDAC2NCOR2
SCHEMBL22563014 0.75 MAPK1 (0.34) HDAC1
SCHEMBL22564663 0.73 HDAC1 (0.34) HDAC1HDAC3HDAC2NCOR2
SCHEMBL22563056 0.71 HDAC1 (0.41) HDAC1HDAC3HDAC2NCOR2
SCHEMBL22564672 0.70 HDAC1 (0.35) HDAC1
SCHEMBL22564671 0.68 HDAC8 (0.34) HDAC1HDAC3HDAC2ITGB3NCOR2
SCHEMBL22562991 0.61 RARB (0.49)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3725777-A1 BENZO- AND PYRIDO-PYRAZOLES AS PROTEIN KINASE INHIBITORS Rottapharm Biotech S.r.l. (IT) 2020-10-21 EP disclosed