SCHEMBL2256346

SCHEMBL2256346

Nc1cccc2[c]cccc12

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.55
CYP3A4 P08684 5/20 0.55
HPGD P15428 4/20 0.55
TSHR P16473 3/20 0.55
HSD17B10 Q99714 2/20 0.55
TDP1 Q9NUW8 2/20 0.55
KEAP1 Q14145 2/20 0.46
NR4A2 P43354 2/20 0.43
ALOX15 P16050 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
KDM4E B2RXH2 3/20 0.39
KMT2A Q03164 3/20 0.39
LMNA P02545 3/20 0.39
MEN1 O00255 2/20 0.39
MAPT P10636 2/20 0.39
GAA P10253 2/20 0.39
PARP1 P09874 2/20 0.36
IDO1 P14902 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL249412 0.83 ALDH1A1 (0.43) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL2333542 0.83 ALDH1A1 (0.43) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL2318595 0.78 CYP1A2 (0.32) CYP1A2
SCHEMBL7295227 0.77 MEN1 (0.39) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL2411016 0.76 CYP1A2 (0.32) CYP1A2
SCHEMBL386156 0.76 CYP1A2 (0.55) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL2252554 0.76 ALDH1A1 (0.42) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL2251412 0.76 ALDH1A1 (0.42) ALDH1A1CYP3A4HPGDTSHRHSD17B10
SCHEMBL4166774 0.74 NOS1 (0.32)
SCHEMBL386939 0.74 HSD17B10 (0.44) ALDH1A1CYP3A4HPGDTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 75 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1434763-B1 BETA-LACTAMYL VASOPRESSIN V1A ANTAGONISTS AZEVAN PHARMACEUTICALS INC (US) 2018-01-17 EP disclosed
CN-104826290-B The golf of layer composition is covered with photostability and durability 阿库施耐特公司 2017-06-23 CN disclosed
CN-105833483-A Multi-piece golf ball comprising low hardness gradient core 阿库施耐特公司 2016-08-10 CN disclosed
CN-102526990-B Comprise the double-core golf of zero gradient center and positive gradient outer nuclear layer 阿库施耐特公司 2016-08-03 CN disclosed
CN-102526994-B Multi-piece golf balls including low hardness gradient cores 阿库施耐特公司 2016-06-08 CN disclosed
US-9006225-B2 Stable pharmaceutical composition ASAHI KASEI PHARMA CORPORATION (JP) 2015-04-14 US disclosed
EP-1916244-B1 THIOPHENE COMPOUND HAVING SULFONYL GROUP AND PROCESS FOR PRODUCING THE SAME NISSAN CHEMICAL IND LTD (JP) 2013-12-04 EP disclosed
CN-101282959-B Thiophene compound having sulfonyl group and method for producing same NISSAN CHEMICAL IND LTD 2013-04-17 CN disclosed
EP-1882694-B1 OLIGOMERS AND POLYMERS OF THIOPHENE COMPOUNDS HAVING PHOSPHORIC ESTER AND PROCESS FOR PRODUCING THE SAME NISSAN CHEMICAL IND LTD (JP) 2013-04-03 EP disclosed
US-8030438-B2 Thiophene compound having phosphoric ester and process for producing the same NISSAN CHEMICAL INDUSTRIES, LTD. (JP) 2011-10-04 US disclosed
EP-0653066-A1 PHOTOACTIVATABLE CHEMILUMINESCENT MATRICES BEHRINGWERKE Aktiengesellschaft (DE) 1995-05-17 EP disclosed
US-5391556-A Thrombin inhibitors KARL THOMAE GMBH (DE) 1995-02-21 US disclosed
US-5340716-A Assay method utilizing photoactivated chemiluminescent label SNYTEX (U.S.A.) INC. (US) 1994-08-23 US disclosed
WO-1994003812-A1 PHOTOACTIVATABLE CHEMILUMINESCENT MATRICES SYNTEX (U.S.A.) INC. (US) 1994-02-17 WO disclosed
EP-0555824-A1 N-alpha-arylsulfonylated benzimidazolylalaninamide derivatives, medicaments based thereon and process for their preparation Dr. Karl Thomae GmbH (DE) 1993-08-18 EP disclosed
EP-0515194-A2 Assay methods utilizing induced luminescence BEHRINGWERKE Aktiengesellschaft (DE) 1992-11-25 EP disclosed
US-4818814-A COLORFASTNESS HOECHST AKTIENGESELLSCHAFT (DE) 1989-04-04 US disclosed
EP-0027906-B1 PROCESS FOR PREPARING SULPHON AMIDES BAYER AG (DE) 1983-05-25 EP disclosed
US-4322214-A USING A SULFUR OR SULFURIZED VAT DYE IN AN ALKALINE BATH CONTAINING A MERCAPTO COMPOUND AND A SULFITE SALT; LEVELING ASAHI CHEMICAL COMPANY LIMITED (JP) 1982-03-30 US disclosed
EP-0027906-A1 Process for preparing sulphon amides BAYER AG (DE) 1981-05-06 EP disclosed