SCHEMBL22600407

SCHEMBL22600407

CC(C)c1cn(C)c(=O)c2[nH]ncc12

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
METAP2 P50579 7/20 0.36
BRD4 O60885 6/20 0.35
KDM5A P29375 1/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM5B Q9UGL1 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22600170 0.76 BRD4 (0.40) METAP2BRD4ALDH1A1KDM4EHPGD
SCHEMBL15069186 0.76 BRD4 (0.37) METAP2BRD4ALDH1A1KDM4EHPGD
SCHEMBL21445298 0.73 BRD4 (0.55) BRD4
SCHEMBL12258192 0.71 HSP90AA1 (0.41) HSP90AA1HSP90AB1METAP2ALDH1A1KDM4E
SCHEMBL23589864 0.70 BRD9 (0.43) METAP2BRD4ALDH1A1KDM4EHPGD
SCHEMBL29303306 0.70 LMNA (0.39) BRD4ALDH1A1HPGD
SCHEMBL24556359 0.69 BRD4 (0.43) BRD4
SCHEMBL24556402 0.69 BRD4 (0.44) BRD4
SCHEMBL12563121 0.68 BRD4 (0.55) BRD4ALDH1A1
SCHEMBL19297126 0.68 HSP90AA1 (0.37) HSP90AA1HSP90AB1METAP2ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020219168-A1 SMALL MOLECULE BROMODOMAIN INHIBITORS AND USES THEREOF CONVERGENE, LLC (US) 2020-10-29 WO disclosed