SCHEMBL22607376

SCHEMBL22607376

Cc1cc(-c2cccn2C)cc(C(C)C)c1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.40
CYP2A6 P11509 1/20 0.40
CYP2A13 Q16696 1/20 0.40
EPHX2 P34913 1/20 0.39
PCSK9 Q8NBP7 1/20 0.38
KDM4E B2RXH2 3/20 0.34
GAA P10253 2/20 0.34
HTT P42858 1/20 0.33
JAK2 O60674 2/20 0.32
ALOX15 P16050 1/20 0.31
BRD9 Q9H8M2 1/20 0.31
BRD7 Q9NPI1 1/20 0.31
LMNA P02545 1/20 0.31
SLC6A3 Q01959 1/20 0.31
NPC1 O15118 1/20 0.30
RECQL P46063 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18999650 0.90 PCSK9 (0.46) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL19007341 0.84 ALDH1A1 (0.48) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL24992270 0.80 ALDH1A1 (0.37) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL26529342 0.77 PCSK9 (0.47) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL17127671 0.73 ALDH1A1 (0.40) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL28310880 0.70 PCSK9 (0.52) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL11951635 0.70 LMNA (0.47) ALDH1A1CYP2A6CYP2A13PCSK9KDM4E
SCHEMBL6067863 0.67 ALDH1A1 (0.47) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL197196 0.66 PCSK9 (0.60) ALDH1A1CYP2A6CYP2A13EPHX2PCSK9
SCHEMBL3363012 0.66 LMNA (0.40) ALDH1A1CYP2A6KDM4EGAAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3122353-B1 SUBSTITUTED INDOLE MCL-1 INHIBITORS UNIV VANDERBILT (US) 2020-10-28 EP disclosed