SCHEMBL22608957

SCHEMBL22608957

COc1ccc2nc3[nH]nc(C)c3c(NC(C)OCCO)c2c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.50
AURKA O14965 1/20 0.40
CDK1 P06493 1/20 0.40
CDK4 P11802 1/20 0.40
CDK2 P24941 1/20 0.40
AKT1 P31749 1/20 0.40
KCNH2 Q12809 2/20 0.39
ADORA2A P29274 1/20 0.38
HSD17B10 Q99714 5/20 0.37
KDM4E B2RXH2 5/20 0.37
ALDH1A1 P00352 4/20 0.37
POLB P06746 3/20 0.37
HPGD P15428 3/20 0.37
MEN1 O00255 5/20 0.36
KMT2A Q03164 5/20 0.36
USP2 O75604 4/20 0.36
TP53 P04637 3/20 0.36
CYP3A4 P08684 3/20 0.36
CASP1 P29466 3/20 0.36
CASP7 P55210 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18079552 0.75 AURKA (0.52) NUDT1AURKACDK1CDK4CDK2
SCHEMBL9006232 0.73 AURKA (0.50) NUDT1AURKACDK1CDK4CDK2
SCHEMBL15574808 0.72 NUDT1 (0.60) NUDT1AURKACDK1CDK4CDK2
SCHEMBL15574603 0.71 NUDT1 (0.60) NUDT1AURKACDK1CDK4CDK2
SCHEMBL9006329 0.71 NUDT1 (0.41) NUDT1AURKACDK1CDK4CDK2
SCHEMBL9006085 0.71 POLB (0.49) NUDT1AURKACDK1CDK4CDK2
SCHEMBL9006179 0.71 PPARA (0.46) NUDT1AURKACDK1CDK4CDK2
SCHEMBL9006315 0.69 AURKA (0.46) NUDT1AURKACDK1CDK4CDK2
SCHEMBL9006235 0.67 HPGD (0.49) AURKACDK1CDK4CDK2AKT1
SCHEMBL29911258 0.67 NUDT1 (1.00) NUDT1AURKACDK1CDK4CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3733840-A1 PLURIPOTENT STEM CELL AGGREGATION INHIBITOR Kaneka Corporation (JP) 2020-11-04 EP disclosed