Romifidine

Romifidine

SCHEMBL22616282

Fc1cccc(Br)c1NC1=NCCN1.O=C(O)C(F)(F)F

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 9/20 0.46
ADRA2C P18825 8/20 0.46
ADRA2B P18089 7/20 0.46
ADRA1A P35348 4/20 0.46
ADRA1D P25100 3/20 0.46
ADRA1B P35368 3/20 0.46
HTR1D P28221 3/20 0.46
LMNA P02545 2/20 0.46
MEN1 O00255 1/20 0.46
SLC22A1 O15245 1/20 0.46
SLC22A3 O75751 1/20 0.46
HTR1A P08908 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
HRH2 P25021 1/20 0.46
CYP2C19 P33261 1/20 0.46
OPRK1 P41145 1/20 0.46
KMT2A Q03164 1/20 0.46
HIF1A Q16665 1/20 0.46
SLC47A1 Q96FL8 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Romifidine SCHEMBL22616289 1.00 ADRA2A (0.46) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616243 0.92 ADRA2A (0.43) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616264 0.92 ADRA2A (0.43) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616132 0.90 ADRA2A (0.41) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616310 0.89 HTR1D (0.50) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL29761110 0.89 ADRA2C (0.56) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL246009 0.89 ADRA2C (0.56) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616245 0.88 HTR1D (0.52) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616284 0.87 ADRA2C (0.55) ADRA2AADRA2CADRA2BADRA1AADRA1D
Romifidine SCHEMBL1970327 0.87 ADRA2C (0.57) ADRA2AADRA2CADRA2BADRA1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220211672-A1 METHODS OF TREATING PRURITUS CLEXIO BIOSCIENCES LTD. (IL) 2022-07-07 US disclosed
WO-2020222192-A1 METHODS OF TREATING PRURITUS CLEXIO BIOSCIENCES LTD. (IL) 2020-11-05 WO disclosed