Romifidine

Romifidine

SCHEMBL246009

Fc1cccc(Br)c1NC1=NCCN1

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2C P18825 13/20 0.56
ADRA2A P08913 12/20 0.56
ADRA2B P18089 12/20 0.56
ADRA1A P35348 5/20 0.56
ADRA1D P25100 4/20 0.56
ADRA1B P35368 4/20 0.56
HTR1D P28221 3/20 0.56
LMNA P02545 2/20 0.56
CYP2D6 P10635 2/20 0.56
NISCH Q9Y2I1 2/20 0.56
MEN1 O00255 1/20 0.56
SLC22A1 O15245 1/20 0.56
SLC22A3 O75751 1/20 0.56
HTR1A P08908 1/20 0.56
CYP2C9 P11712 1/20 0.56
HRH2 P25021 1/20 0.56
CYP2C19 P33261 1/20 0.56
OPRK1 P41145 1/20 0.56
KMT2A Q03164 1/20 0.56
HIF1A Q16665 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Romifidine SCHEMBL29761110 1.00 ADRA2C (0.56) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL1970327 0.98 ADRA2C (0.57) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616284 0.98 ADRA2C (0.55) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616255 0.92 ADRA2C (0.49) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616210 0.92 ADRA2C (0.49) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616229 0.91 ADRA2C (0.48) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616310 0.90 HTR1D (0.50) ADRA2CADRA2AADRA2BADRA1AADRA1D
SCHEMBL11182818 0.89 ADRA2C (0.65) ADRA2CADRA2AADRA2BADRA1AADRA1D
SCHEMBL9920134 0.89 ADRA2C (0.65) ADRA2CADRA2AADRA2BADRA1AADRA1D
Romifidine SCHEMBL22616282 0.89 ADRA2A (0.46) ADRA2CADRA2AADRA2BADRA1AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 710 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4704839-A2 IMIDAZOLE CONTAINING COMPOUNDS, DERIVATIVES THEREFORE, AND USES THEREOF ALPHERABIO LLC (US) 2026-03-11 EP claimed
US-12501899-B2 Mite infestation treatment VETO-PHARMA (FR) 2025-12-23 US claimed
EP-4661680-A1 COMPOSITION FOR CONTROLLING MITE INFESTATION Veto-Pharma (FR) 2025-12-17 EP claimed
WO-2025080559-A1 METHODS AND COMPOSITIONS FOR TREATING DRUG OVERDOSE ENALARE THERAPEUTICS INC. (US) 2025-04-17 WO claimed
US-20250114370-A1 METHODS AND COMPOSITIONS FOR TREATING DRUG OVERDOSE ENALARE THERAPEUTICS INC (US) 2025-04-10 US claimed
WO-2024226608-A2 IMIDAZOLE CONTAINING COMPOUNDS, DERIVATIVES THEREFORE, AND USES THEREOF AGLAEAPHARMA INC. (US) 2024-10-31 WO claimed
WO-2024165712-A1 COMPOSITION FOR CONTROLLING MITE INFESTATION VETO-PHARMA (FR) 2024-08-15 WO claimed
EP-4413861-A1 COMPOSITION FOR CONTROLLING MITE INFESTATION Veto-Pharma (FR) 2024-08-14 EP claimed
US-20240139181-A1 METHODS FOR INDUCING PUPIL DILATION THE REGENTS OF THE UNIVERSITY OF COLORADO, A BODY CORPORATE 2024-05-02 US claimed
US-20230404979-A1 ALPHA-2 ADRENERGIC RECEPTOR AGONISTS TO REDUCE MORTALITY AND IMPROVE OUTCOMES IN VIRAL RESPIRATORY SYNDROMES RUSH UNIVERSITY MEDICAL CENTER (US) 2023-12-21 US claimed
WO-2007061529-A1 LYOPHILIZATION PROCESS AND PRODUCTS OBTAINED THEREBY SCIDOSE LLC. (US) 2007-05-31 WO claimed
US-20070116729-A1 Lyophilization process and products obtained thereby SCIDOSE LLC 2007-05-24 US claimed
EP-1273301-B1 Pharmaceutical preparations based on active ingredients susceptible to illicit administration ALTERGON SA (CH) 2006-09-06 EP claimed
EP-1273301-A2 Pharmaceutical preparations based on active ingredients susceptible to illicit administration ALTERGON S.A. (CH) 2003-01-08 EP claimed
EP-0719139-A1 USE OF CENTRALLY ACTIVE ALPHAAGONISTS FOR INHIBING POSTRAUMATIC METABOLIC STRESS Dr. Karl Thomae GmbH (DE) 1996-07-03 EP claimed
WO-1995003798-A2 USE OF CENTRALLY EFFECTIVE α-2 AGONISTS FOR INHIBITING POSTAGGRESSION METABOLISM BOEHRINGER INGELHEIM INT (DE) 1995-02-09 WO claimed
EP-0170193-B1 FEEDSTUFF ADDITIVE FOR THE GROWTH PROMOTING OF AGRICULTURAL USEFUL ANIMALS BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 1991-12-27 EP claimed
US-4853402-A 2-SUBSTITUTED-2-IMIDAZOLINES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 1989-08-01 US claimed
EP-0170193-A2 Feedstuff additive for the growth promoting of agricultural useful animals BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 1986-02-05 EP claimed
EP-0031429-B1 2-(N-(2-FLUORO-6-BROMOPHENYL)-N-(THIEMYL-2-METHYL)-AMINO)-2-IMIDAZOLINE, ITS ADDITION SALTS, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND PROCESSES FOR THEIR PREPARATION C.H. BOEHRINGER SOHN (DE) 1984-07-04 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12501899-B2 Mite infestation treatment RHOA, NPEPPS, TUBA3E ADRA2C 2479/4885ADRA2A 3402/4885ADRA2B 3269/4885
US-20250114370-A1 METHODS AND COMPOSITIONS FOR TREATING DRUG OVERDOSE ADRA2A, ADRA2C, OPRM1 ADRA2C 2/4885ADRA2A 1/4885ADRA2B 6/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.