SCHEMBL22628802

SCHEMBL22628802

CC([C@H](C)CN[C@@H](CO)C(=O)O)C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRN P28799 1/20 0.38
SORT1 Q99523 1/20 0.38
TGFBR1 P36897 3/20 0.36
MME P08473 5/20 0.35
PDCD1 Q15116 1/20 0.31
CD274 Q9NZQ7 1/20 0.31
MAPT P10636 1/20 0.31
FOLH1 Q04609 2/20 0.31
NAALAD2 Q9Y3Q0 2/20 0.31
ALDH1A1 P00352 1/20 0.31
ACE P12821 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23052826 0.80 TGFBR1 (0.41) TGFBR1MMEMAPTFOLH1NAALAD2
SCHEMBL21451281 0.75 MME (0.46) TGFBR1MMEMAPTFOLH1NAALAD2
SCHEMBL21451346 0.75 MME (0.46) TGFBR1MMEMAPTFOLH1NAALAD2
SCHEMBL23052781 0.75 MME (0.46) TGFBR1MMEMAPTFOLH1NAALAD2
SCHEMBL18822312 0.70 CTSS (0.44) GRNSORT1TGFBR1MMEPDCD1
SCHEMBL22487801 0.69 TGFBR1 (0.47) TGFBR1MMEPDCD1CD274MAPT
SCHEMBL30925323 0.69 TGFBR1 (0.39) TGFBR1MMEMAPTFOLH1NAALAD2
SCHEMBL13395755 0.68 TSHR (0.37)
SCHEMBL13395757 0.68 TSHR (0.37)
SCHEMBL13395730 0.68 TSHR (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3733659-A1 AROMATIC VINYL OR AROMATIC ETHYL DERIVATIVE, PREPARATION METHOD THEREFOR, INTERMEDIATE, PHARMACEUTICAL COMPOSITION, AND APPLICATION Guangzhou Maxinovel Pharmaceuticals Co., Ltd. (CN) 2020-11-04 EP disclosed