SCHEMBL2264146

SCHEMBL2264146

Cc1[c]ccc(Oc2ccc(C)cc2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TEAD4 Q15561 1/20 0.47
ALDH1A1 P00352 3/20 0.45
TDP1 Q9NUW8 2/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
AR P10275 2/20 0.41
HTT P42858 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
PDE4A P27815 1/20 0.38
PDE4B Q07343 1/20 0.38
PDE4C Q08493 1/20 0.38
PDE4D Q08499 1/20 0.38
ACHE P22303 1/20 0.38
MMP13 P45452 2/20 0.38
LPAR1 Q92633 1/20 0.36
LPAR3 Q9UBY5 1/20 0.36
HSD17B1 P14061 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1375387 0.85 SOS1 (0.38) ALDH1A1SMN1; SMN2PDE4APDE4BPDE4C
SCHEMBL1584803 0.84 LTA4H (0.48) ALDH1A1TDP1MAPTHTTL3MBTL1
SCHEMBL5583787 0.82 TEAD4 (0.45) TEAD4ALDH1A1TDP1POLBMAPT
SCHEMBL21630305 0.81 TEAD4 (0.44) TEAD4ALDH1A1TDP1POLBMAPT
SCHEMBL920492 0.81 TEAD4 (0.44) TEAD4ALDH1A1TDP1POLBMAPT
SCHEMBL14937866 0.80 SLC6A4 (0.37) POLBMAPTARL3MBTL1PTGS2
SCHEMBL5583736 0.77 AR (0.51) TEAD4ALDH1A1TDP1POLBMAPT
SCHEMBL921069 0.76 TEAD4 (0.56) TEAD4ALDH1A1TDP1POLBMAPT
SCHEMBL20243511 0.76 GRM5 (0.35) TDP1CYP2C9CYP3A4
SCHEMBL83814 0.75 TEAD4 (0.74) TEAD4ALDH1A1TDP1POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7998986-B2 Heterocyclic compounds, in particular N-substituted pyridones for modulating the activity of nuclear receptors EXELIXIS PATENT COMPANY LLC (US) 2011-08-16 US claimed