SCHEMBL22650422

SCHEMBL22650422

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCCNC5=O)cc4)n3)cc12

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK1 P06493 3/20 0.41
CCNB1 P14635 3/20 0.41
CDK2 P24941 2/20 0.41
CCNA2 P20248 1/20 0.41
CCNA1 P78396 1/20 0.41
STK17A Q9UEE5 5/20 0.40
MYLK4 Q86YV6 4/20 0.40
JAK2 O60674 10/20 0.40
CDK4 P11802 2/20 0.39
CCND1 P24385 2/20 0.39
NEK3 P51956 1/20 0.38
LIMK1 P53667 1/20 0.38
NEK5 Q6P3R8 1/20 0.38
CDK6 Q00534 1/20 0.38
JAK3 P52333 4/20 0.38
ABL1 P00519 1/20 0.38
PDGFRB P09619 1/20 0.38
BCR P11274 1/20 0.38
SRC P12931 1/20 0.38
PDGFRA P16234 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650366 0.90 CDK4 (0.47) CDK1CCNB1CDK2CCNA2CCNA1
SCHEMBL22650526 0.87 MAP4K1 (0.44) CDK1CCNB1CDK2CCNA2CCNA1
SCHEMBL22650707 0.86 JAK2 (0.39) CDK1CCNB1STK17AMYLK4JAK2
SCHEMBL22650709 0.86 JAK2 (0.39) CDK1CCNB1STK17AMYLK4JAK2
SCHEMBL22650924 0.85 CDK4 (0.48) CDK1CCNB1CDK2CCNA2CCNA1
SCHEMBL22650419 0.84 JAK2 (0.38) CDK1CCNB1STK17AMYLK4JAK2
SCHEMBL22650847 0.83 JAK2 (0.39) CDK1CCNB1CDK2CCNA2CCNA1
SCHEMBL22650766 0.82 JAK2 (0.39) CDK1CCNB1CDK2CCNA2CCNA1
SCHEMBL22650421 0.81 JAK2 (0.38) CDK1CCNB1CDK2CCNA2CCNA1
SCHEMBL22650921 0.80 MTOR (0.49) CDK1CCNB1CDK2STK17AMYLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed