SCHEMBL22650709

SCHEMBL22650709

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCCC(N)C5=O)cc4)n3)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 9/20 0.39
JAK3 P52333 6/20 0.39
CDK9 P50750 5/20 0.38
BRD4 O60885 3/20 0.38
ABL1 P00519 1/20 0.38
PDGFRB P09619 1/20 0.38
BCR P11274 1/20 0.38
SRC P12931 1/20 0.38
PDGFRA P16234 1/20 0.38
PRKCA P17252 1/20 0.38
PRKCD Q05655 1/20 0.38
CDK1 P06493 1/20 0.37
CDK4 P11802 1/20 0.37
CCNB1 P14635 1/20 0.37
CCND1 P24385 1/20 0.37
STK17A Q9UEE5 3/20 0.37
MYLK4 Q86YV6 2/20 0.37
NEK3 P51956 1/20 0.37
LIMK1 P53667 1/20 0.37
NEK5 Q6P3R8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650707 0.91 JAK2 (0.39) JAK2JAK3CDK9BRD4CDK1
SCHEMBL22650419 0.89 JAK2 (0.38) JAK2JAK3CDK9BRD4CDK1
SCHEMBL22650519 0.89 EGFR (0.36) CDK9BRD4ABL1PDGFRBBCR
SCHEMBL22650523 0.88 EGFR (0.42) JAK2CDK5CDK5R1
SCHEMBL22650702 0.88 JAK2 (0.39) JAK2JAK3CDK9BRD4ABL1
SCHEMBL22650847 0.86 JAK2 (0.39) JAK2JAK3CDK9BRD4ABL1
SCHEMBL22650422 0.86 CDK1 (0.41) JAK2JAK3CDK9ABL1PDGFRB
SCHEMBL22650701 0.85 JAK2 (0.38) JAK2JAK3CDK9BRD4ABL1
SCHEMBL22650940 0.83 BTK (0.38) CDK9BRD4CDK1CDK4CCNB1
SCHEMBL22650450 0.83 CDK4 (0.41) CDK9CDK1CDK4CCNB1CCND1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed