SCHEMBL22650424

SCHEMBL22650424

CCN1CCC(Cn2ccc(Nc3nccc(-c4cc5c(ncn5C(C)C)c(OC)n4)n3)n2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 5/20 0.39
CDK6 Q00534 5/20 0.35
CCND1 P24385 4/20 0.35
LRRK2 Q5S007 2/20 0.34
CDK4 P11802 4/20 0.34
CDK1 P06493 3/20 0.34
CCND3 P30281 3/20 0.34
CCNT1 O60563 3/20 0.33
CDK9 P50750 3/20 0.33
CCNB1 P14635 2/20 0.33
CCNA2 P20248 2/20 0.33
CDK2 P24941 2/20 0.33
CDK7 P50613 2/20 0.33
CCNH P51946 2/20 0.33
CCNE1 P24864 1/20 0.33
ZAP70 P43403 2/20 0.33
ACVR1 Q04771 1/20 0.32
AURKA O14965 1/20 0.32
LCK P06239 1/20 0.32
KDR P35968 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650473 0.90 MAP3K14 (0.41) MAP3K14LRRK2CCNA2CDK2CCNE1
SCHEMBL22650429 0.75 CCND1 (0.40) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650946 0.75 CDK6 (0.44) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650856 0.74 CDK6 (0.47) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650860 0.73 CDK6 (0.44) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650511 0.72 CCND1 (0.35) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650859 0.72 CDK4 (0.51) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650734 0.72 CDK6 (0.48) CDK6CCND1CDK4CDK1CCND3
SCHEMBL22650407 0.67 L3MBTL1 (0.37) CDK1CCNA2CDK2
SCHEMBL22650503 0.67 MAPK14 (0.46) MAP3K14CDK1CCNT1CDK9CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed