SCHEMBL22650473

SCHEMBL22650473

COc1nc(-c2ccnc(Nc3ccn(CC4CCNCC4)n3)n2)cc2c1ncn2C(C)C

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 6/20 0.41
LRRK2 Q5S007 3/20 0.35
TGFBR1 P36897 1/20 0.34
BRD4 O60885 2/20 0.33
ALK Q9UM73 1/20 0.33
MAP3K5 Q99683 1/20 0.33
EGFR P00533 1/20 0.32
CCNE2 O96020 1/20 0.32
CCNA2 P20248 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
CCNA1 P78396 1/20 0.32
MKNK1 Q9BUB5 1/20 0.32
MKNK2 Q9HBH9 1/20 0.32
BRD2 P25440 1/20 0.32
BRD3 Q15059 1/20 0.32
BRDT Q58F21 1/20 0.32
ACVR1 Q04771 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650424 0.90 MAP3K14 (0.39) MAP3K14LRRK2MAP3K5EGFRCCNA2
SCHEMBL22650775 0.75 CDK4 (0.44) CCNA2CDK2
SCHEMBL22650489 0.73 MAP3K14 (0.48) MAP3K14LRRK2CCNA2CCNE1CDK2
SCHEMBL22650946 0.72 CDK6 (0.44) EGFRCCNE2CCNA2CCNE1CDK2
SCHEMBL22650856 0.71 CDK6 (0.47) CCNA2CDK2CCNA1
SCHEMBL22650859 0.70 CDK4 (0.51) CCNA2CDK2CCNA1
SCHEMBL22650734 0.70 CDK6 (0.48) CCNA2CDK2CCNA1
SCHEMBL22650549 0.69 ZAP70 (0.42) EGFRCCNA2CDK2CCNA1ACVR1
SCHEMBL22650503 0.68 MAPK14 (0.46) MAP3K14CCNA2CCNE1CDK2CCNA1
SCHEMBL22650407 0.68 L3MBTL1 (0.37) CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed