SCHEMBL22650430

SCHEMBL22650430

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCNCC5=O)nc4)n3)cc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MYLK4 Q86YV6 2/20 0.43
STK17A Q9UEE5 2/20 0.43
CLK4 Q9HAZ1 1/20 0.43
TBK1 Q9UHD2 1/20 0.43
ZAP70 P43403 6/20 0.41
PRKD3 O94806 1/20 0.41
EGFR P00533 1/20 0.41
PRKCG P05129 1/20 0.41
PRKCB P05771 1/20 0.41
LCK P06239 1/20 0.41
PRKCA P17252 1/20 0.41
PRKCH P24723 1/20 0.41
PRKCI P41743 1/20 0.41
PRKCE Q02156 1/20 0.41
PRKCQ Q04759 1/20 0.41
PRKCZ Q05513 1/20 0.41
PRKCD Q05655 1/20 0.41
PRKD1 Q15139 1/20 0.41
ACVR1 Q04771 2/20 0.37
IKBKB O14920 5/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650526 0.91 MAP4K1 (0.44) MYLK4STK17AIKBKBCHUKCDK1
SCHEMBL22650426 0.88 IKBKB (0.42) ACVR1IKBKBCHUKCDK1CCNB1
SCHEMBL22650939 0.88 CAMK2D (0.44) STK17AEGFRPRKCAPRKCDIKBKB
SCHEMBL29491175 0.85 CDK4 (0.49) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL22650568 0.85 CDK4 (0.49) CDK1CCNB1CCNA2CDK2CCNA1
SCHEMBL22650937 0.84 CDK4 (0.40) MYLK4STK17AEGFRCDK1CCNB1
SCHEMBL22650432 0.83 CDK6 (0.35) ZAP70PRKD3EGFRPRKCGPRKCB
SCHEMBL22650524 0.83 CDK6 (0.38) MYLK4STK17AEGFRIKBKBCHUK
SCHEMBL22650940 0.82 BTK (0.38) MYLK4STK17ACLK4TBK1ZAP70
SCHEMBL22650485 0.81 CDK4 (0.47) CDK1CCNB1CCNA2CDK2CCNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed