SCHEMBL22650432

SCHEMBL22650432

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCNCC5=O)c(F)c4F)n3)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 5/20 0.35
CDK4 P11802 4/20 0.35
CDK1 P06493 2/20 0.35
CCNB1 P14635 1/20 0.35
CCND1 P24385 1/20 0.35
CSF1R P07333 1/20 0.35
IKBKB O14920 2/20 0.34
MAP3K14 Q99558 2/20 0.34
MAPK1 P28482 5/20 0.33
MAPK3 P27361 3/20 0.33
SOS1 Q07889 1/20 0.33
PIK3CG P48736 3/20 0.32
MAPK8 P45983 2/20 0.32
CAMKK2 Q96RR4 2/20 0.32
GSK3B P49841 1/20 0.32
CHUK O15111 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
CCND3 P30281 2/20 0.32
EGFR P00533 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650524 0.90 CDK6 (0.38) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650426 0.88 IKBKB (0.42) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650937 0.86 CDK4 (0.40) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650526 0.84 MAP4K1 (0.44) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650430 0.83 MYLK4 (0.43) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL29491175 0.83 CDK4 (0.49) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650568 0.83 CDK4 (0.49) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650939 0.82 CAMK2D (0.44) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650485 0.79 CDK4 (0.47) CDK6CDK4CDK1CCNB1CCND1
SCHEMBL22650922 0.78 F10 (0.38) MAP3K14MAPK8EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed