SCHEMBL22650454

SCHEMBL22650454

CC(C)(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5C(=O)C6CC5CN6)cn4)n3)cc12

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 17/20 0.39
CCND1 P24385 13/20 0.39
CDK6 Q00534 11/20 0.39
CDK1 P06493 8/20 0.39
CCNB1 P14635 6/20 0.39
CCNA2 P20248 10/20 0.36
CCND3 P30281 9/20 0.36
CDK2 P24941 10/20 0.36
CCNE1 P24864 5/20 0.36
CCNA1 P78396 5/20 0.33
CCNT1 O60563 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
CCNH P51946 1/20 0.32
MNAT1 P51948 1/20 0.32
CDK5 Q00535 1/20 0.32
CDK5R1 Q15078 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650449 0.88 CDK4 (0.42) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650521 0.79 CDK4 (0.40) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650527 0.79 CDK4 (0.40) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650763 0.78 CDK4 (0.47) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650705 0.77 CDK6 (0.39) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650702 0.71 JAK2 (0.39) CCNA2CDK2CCNA1CDK9
SCHEMBL22650924 0.69 CDK4 (0.48) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL22650428 0.69 CDK4 (0.35) CDK4CDK6CDK1CCNA2CCND3
SCHEMBL22650366 0.68 CDK4 (0.47) CDK4CCND1CDK6CDK1CCNB1
SCHEMBL29491175 0.67 CDK4 (0.49) CDK4CCND1CDK6CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed