SCHEMBL22650702

SCHEMBL22650702

CC(C)(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCCC(N)C5=O)cc4)n3)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 9/20 0.39
JAK3 P52333 5/20 0.39
ABL1 P00519 2/20 0.38
BCR P11274 2/20 0.38
SRC P12931 2/20 0.38
PDGFRB P09619 1/20 0.38
PDGFRA P16234 1/20 0.38
PRKCA P17252 1/20 0.38
PRKCD Q05655 1/20 0.38
STK17A Q9UEE5 2/20 0.37
BTK Q06187 3/20 0.36
BRD4 O60885 1/20 0.36
CDK9 P50750 1/20 0.36
MAPK10 P53779 1/20 0.36
JAK1 P23458 1/20 0.36
MYLK4 Q86YV6 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
CCNA1 P78396 1/20 0.36
EGFR P00533 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650521 0.91 CDK4 (0.40) CDK9CCNA2CDK2
SCHEMBL22650428 0.89 CDK4 (0.35) ABL1BCRPDGFRBBTKBRD4
SCHEMBL22650709 0.88 JAK2 (0.39) JAK2JAK3ABL1BCRSRC
SCHEMBL22650527 0.83 CDK4 (0.40) BTKCDK9CCNA2CDK2CCNA1
SCHEMBL22650701 0.81 JAK2 (0.38) JAK2JAK3ABL1BCRSRC
SCHEMBL22650707 0.79 JAK2 (0.39) JAK2JAK3STK17ABTKBRD4
SCHEMBL22650419 0.77 JAK2 (0.38) JAK2JAK3STK17ABRD4CDK9
SCHEMBL22650519 0.77 EGFR (0.36) ABL1BCRPDGFRBBRD4CDK9
SCHEMBL22650523 0.77 EGFR (0.42) JAK2CDK2EGFR
SCHEMBL22650847 0.74 JAK2 (0.39) JAK2JAK3ABL1BCRSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed