SCHEMBL22650521

SCHEMBL22650521

CC(C)(C)c1cnn2ccc(-c3ccnc(Nc4ccc(N5CCCC(N)C5=O)cn4)n3)cc12

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 18/20 0.40
CDK6 Q00534 15/20 0.40
CCND3 P30281 13/20 0.40
CCND1 P24385 10/20 0.39
CDK1 P06493 9/20 0.39
CCNB1 P14635 7/20 0.39
CCNA2 P20248 9/20 0.38
CDK2 P24941 8/20 0.37
CCNT1 O60563 6/20 0.37
CDK9 P50750 6/20 0.37
CDK7 P50613 5/20 0.37
CCNH P51946 5/20 0.37
CCNE1 P24864 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650702 0.91 JAK2 (0.39) CCNA2CDK2CDK9
SCHEMBL22650527 0.90 CDK4 (0.40) CDK4CDK6CCND3CCND1CDK1
SCHEMBL22650428 0.88 CDK4 (0.35) CDK4CDK6CCND3CDK1CCNA2
SCHEMBL22650705 0.83 CDK6 (0.39) CDK4CDK6CCND3CCND1CDK1
SCHEMBL22650763 0.81 CDK4 (0.47) CDK4CDK6CCND3CCND1CDK1
SCHEMBL22650454 0.79 CDK4 (0.39) CDK4CDK6CCND3CCND1CDK1
SCHEMBL22650709 0.79 JAK2 (0.39) CDK4CCND1CDK1CCNB1CDK9
SCHEMBL22650450 0.79 CDK4 (0.41) CDK4CDK6CCND3CCND1CDK1
SCHEMBL22650795 0.78 CDK4 (0.41) CDK4CDK6CCND3CCND1CDK1
SCHEMBL22650519 0.76 EGFR (0.36) CDK4CDK6CCND3CCND1CDK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed