SCHEMBL22650494

SCHEMBL22650494

CC(C)c1cnn2ccc(-c3ccnc(Nc4ccn(CC5CCN(C(=O)CO)CC5)n4)n3)cc12

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAP3K14 Q99558 8/20 0.46
CDK2 P24941 1/20 0.38
IGF1R P08069 1/20 0.37
KCNH2 Q12809 1/20 0.37
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35
MAPK1 P28482 2/20 0.34
BTK Q06187 2/20 0.34
MAPK3 P27361 1/20 0.34
TBK1 Q9UHD2 3/20 0.34
ACVR1 Q04771 1/20 0.34
DYRK2 Q92630 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650461 0.92 MAP3K14 (0.47) MAP3K14JAK2JAK1JAK3TBK1
SCHEMBL22650489 0.86 MAP3K14 (0.48) MAP3K14CDK2TBK1ACVR1
SCHEMBL22650849 0.76 CDK1 (0.47) CDK2JAK2JAK1JAK3DYRK2
SCHEMBL22650848 0.74 CDK1 (0.49) CDK2JAK2JAK1JAK3BTK
SCHEMBL22650936 0.74 IKBKE (0.48) MAP3K14JAK2JAK1JAK3MAPK1
SCHEMBL22650851 0.74 IKBKB (0.56) CDK2
SCHEMBL22650921 0.73 MTOR (0.49) CDK2DYRK2
SCHEMBL22650925 0.73 CDK2 (0.61) CDK2KCNH2JAK1ACVR1
SCHEMBL22650923 0.72 MAPK8 (0.54) CDK2KCNH2JAK2ACVR1
SCHEMBL22650920 0.71 CDK2 (0.54) CDK2KCNH2JAK2JAK1JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed