SCHEMBL22650936

SCHEMBL22650936

CC(C)c1cnn2ccc(-c3ccnc(Nc4cnn(CC5CCNCC5)c4)n3)cc12

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
IKBKE Q14164 12/20 0.48
TBK1 Q9UHD2 12/20 0.48
MYLK4 Q86YV6 2/20 0.43
STK17A Q9UEE5 2/20 0.43
JAK2 O60674 1/20 0.41
JAK1 P23458 1/20 0.41
TYK2 P29597 1/20 0.41
STAT3 P40763 1/20 0.41
JAK3 P52333 1/20 0.41
BTK Q06187 2/20 0.40
MAP3K14 Q99558 1/20 0.40
MAPK3 P27361 1/20 0.38
MAPK1 P28482 1/20 0.38
ACVR1 Q04771 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650489 0.87 MAP3K14 (0.48) IKBKETBK1MAP3K14ACVR1
SCHEMBL22650526 0.75 MAP4K1 (0.44) MYLK4STK17AJAK2JAK3
SCHEMBL22650422 0.74 CDK1 (0.41) MYLK4STK17AJAK2JAK1JAK3
SCHEMBL22650919 0.74 CDK2 (0.54) MYLK4STK17AJAK2JAK3
SCHEMBL22650923 0.74 MAPK8 (0.54) MYLK4STK17AJAK2ACVR1
SCHEMBL22650918 0.74 DKK1 (0.57) JAK2
SCHEMBL22650849 0.74 CDK1 (0.47) MYLK4STK17AJAK2JAK1JAK3
SCHEMBL22650707 0.73 JAK2 (0.39) MYLK4STK17AJAK2JAK3BTK
SCHEMBL22650920 0.73 CDK2 (0.54) MYLK4STK17AJAK2JAK1TYK2
SCHEMBL22650595 0.72 PRKCA (0.40) JAK2JAK3MAP3K14ACVR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed