SCHEMBL22650495

SCHEMBL22650495

CC1(C)COc2c(F)cc(-c3ccnc(Cl)n3)cc21

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.38
KMO O15229 4/20 0.35
PTGS1 P23219 4/20 0.34
PTGS2 P35354 4/20 0.34
ALOX5 P09917 2/20 0.34
MAP3K14 Q99558 3/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
POLB P06746 1/20 0.32
JAK2 O60674 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29462387 1.00 NOTUM (0.38) NOTUMKMOPTGS1PTGS2ALOX5
SCHEMBL28374207 0.71 KMO (0.41) NOTUMKMOALDH1A1
SCHEMBL19836469 0.70 EGFR (0.39) KMO
SCHEMBL30039803 0.70 EGFR (0.39) KMO
SCHEMBL30557503 0.70 CDK4 (0.32)
SCHEMBL29065292 0.70 CDK4 (0.32)
SCHEMBL30557498 0.70 CDK4 (0.34)
SCHEMBL29065294 0.70 CDK4 (0.34)
SCHEMBL16798282 0.70 L3MBTL1 (0.40) KMOALDH1A1
SCHEMBL31375122 0.70 KMO (0.61) KMOPTGS2KDM4EALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114364675-A CDK inhibitors 上海齐鲁锐格医药研发有限公司 2022-04-15 CN disclosed
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed