SCHEMBL22650567

SCHEMBL22650567

COc1cc(N2CCC(N(C)C)CC2=O)ccc1N

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.41
CHEK1 O14757 1/20 0.40
MCHR1 Q99705 2/20 0.39
HTR2A P28223 2/20 0.38
HTR2C P28335 2/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA4 P22748 1/20 0.37
CA7 P43166 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37
ALDH1A1 P00352 2/20 0.37
CYP3A4 P08684 2/20 0.37
TSHR P16473 1/20 0.37
HSD17B10 Q99714 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HSD11B1 P28845 1/20 0.37
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31347314 0.83 BPTF (0.41) HTR2CTSHRHSD11B1POLB
SCHEMBL22650563 0.83 BPTF (0.41) HTR2CTSHRHSD11B1POLB
SCHEMBL310055 0.81 SUV39H2 (0.45) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL29661369 0.81 SUV39H2 (0.45) ALDH1A1CYP3A4TSHRHSD17B10TDP1
Hydrochloric Acid SCHEMBL29367159 0.80 SUV39H2 (0.44) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL22650565 0.79 DDB1 (0.38) ALDH1A1TSHRHSD17B10POLBHTT
SCHEMBL14240636 0.79 NTSR1 (0.47) MCHR1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL520746 0.79 NTSR1 (0.47) MCHR1ALDH1A1CYP3A4TSHRHSD17B10
SCHEMBL20091850 0.75 CHEK1 (0.60) LMNACHEK1ALDH1A1CYP3A4TSHR
SCHEMBL10206636 0.75 ALK (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed