SCHEMBL22650720

SCHEMBL22650720

CC(C)n1cnc2c(F)nc(-c3ccnc(NC4CCN(S(C)(=O)=O)CC4)n3)cc21

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 6/20 0.53
CDK2 P24941 7/20 0.46
CCNE1 P24864 5/20 0.46
CCND1 P24385 11/20 0.46
CDK4 P11802 10/20 0.46
CDK6 Q00534 9/20 0.46
CCND3 P30281 6/20 0.46
CCNT1 O60563 2/20 0.44
CDK9 P50750 2/20 0.44
CDK1 P06493 3/20 0.41
CCNB1 P14635 2/20 0.41
CCNB2 O95067 1/20 0.41
CCNE2 O96020 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41
CCNB3 Q8WWL7 1/20 0.41
MAPK8 P45983 2/20 0.40
MAPK9 P45984 2/20 0.40
MAPK10 P53779 2/20 0.40
CCNA2 P20248 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30874701 0.75 IKBKB (0.68) IKBKBCDK2CCNE1CCND1CDK4
SCHEMBL29212007 0.75 IKBKB (0.68) IKBKBCDK2CCNE1CCND1CDK4
SCHEMBL22650537 0.74 CDK2 (0.50) IKBKBCDK2CCNE1CDK4CCNT1
SCHEMBL22650600 0.71 MAPK14 (0.40) CDK2CDK1CDK5CDK5R1CCNA2
SCHEMBL4504958 0.71 KCNH2 (0.65) IKBKBCDK2CCNE1CCND1CDK4
SCHEMBL30838834 0.71 IKBKB (0.59) IKBKBCDK2CCNE1CCND1CDK4
SCHEMBL29236001 0.71 IKBKB (0.59) IKBKBCDK2CCNE1CCND1CDK4
SCHEMBL22650630 0.71 CDK9 (0.35) CDK2CDK9CDK1CCNB1MAPK10
SCHEMBL22650578 0.71 IKBKB (0.35) IKBKBCDK2CDK9CDK1CCNB1
SCHEMBL22650620 0.71 CDK2 (0.36) CDK2CDK9CDK1CCNB1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed