SCHEMBL22650620

SCHEMBL22650620

CNC1CCCN(c2ccc(Nc3nccc(-c4cc5c(ncn5C(C)C)c(F)n4)n3)cc2)C1=O

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 6/20 0.36
EGFR P00533 1/20 0.35
CDK1 P06493 3/20 0.34
JAK2 O60674 4/20 0.34
JAK3 P52333 3/20 0.34
CDK9 P50750 4/20 0.34
BRD4 O60885 3/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CCNA1 P78396 1/20 0.34
MAPK1 P28482 1/20 0.34
MAP2K1 Q02750 1/20 0.34
KCNH2 Q12809 1/20 0.34
SYK P43405 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650619 0.91 CDK4 (0.40) CDK2CDK1CDK9CCNB1CCNA2
SCHEMBL22650630 0.91 CDK9 (0.35) CDK2EGFRCDK1JAK2JAK3
SCHEMBL22650536 0.89 JAK2 (0.34) CDK2EGFRCDK1JAK2JAK3
SCHEMBL22650535 0.88 CDK2 (0.38) CDK2CDK1JAK2JAK3BRD4
SCHEMBL22650540 0.87 CCND1 (0.40) CDK2EGFR
SCHEMBL22650578 0.86 IKBKB (0.35) CDK2EGFRCDK1JAK2JAK3
SCHEMBL22650626 0.86 CDK2 (0.39) CDK2CDK1JAK2JAK3CDK9
SCHEMBL22650781 0.82 IKBKB (0.39) CDK2EGFRCDK1JAK2JAK3
SCHEMBL22650532 0.81 EGFR (0.36) EGFRCDK9BRD4
SCHEMBL22650777 0.79 ACVR1 (0.35) CDK2EGFRCDK1JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed