SCHEMBL22650757

SCHEMBL22650757

CC(C)n1cnc2c1CN(c1ccnc(Nc3ccc(N4CCCC(N)C4=O)cc3)n1)CC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.35
CCND1 P24385 2/20 0.35
CDK6 Q00534 2/20 0.35
HRH4 Q9H3N8 1/20 0.34
MKNK1 Q9BUB5 2/20 0.34
IDH1 O75874 1/20 0.34
ALK Q9UM73 3/20 0.34
NR2C2 P49116 2/20 0.34
TAB1 Q15750 2/20 0.34
NFKB1 P19838 1/20 0.34
NFKB2 Q00653 1/20 0.34
RELA Q04206 1/20 0.34
JAK2 O60674 8/20 0.33
JAK3 P52333 2/20 0.33
FLT3 P36888 4/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
CCNT1 O60563 1/20 0.33
CCND3 P30281 1/20 0.33
CDK9 P50750 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650753 0.85 CDK4 (0.51) CDK4CCND1CDK6JAK2JAK3
SCHEMBL22650754 0.76 CDK4 (0.51) CDK4CCND1CDK6JAK2JAK3
SCHEMBL22650761 0.76 CDK4 (0.51) CDK4CCND1CDK6JAK2JAK3
SCHEMBL22650444 0.76 CDK4 (0.50) CDK4CCND1CDK6CCNT1CCND3
SCHEMBL22650630 0.73 CDK9 (0.35) JAK2JAK3CDK9CDK1CCNB1
SCHEMBL22650756 0.73 CDK4 (0.44) CDK4CCND1CDK6HRH4CCNT1
SCHEMBL22650765 0.73 CDK4 (0.42) CDK4CCND1CDK6CCNT1CCND3
SCHEMBL22650741 0.72 CDK4 (0.44) CDK4CCND1CDK6JAK2JAK3
SCHEMBL22650552 0.72 CDK4 (0.53) CDK4CCND1CDK6JAK2JAK3
SCHEMBL22650742 0.69 TRPV1 (0.40) CDK4CCND1CDK6HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed