SCHEMBL22650772

SCHEMBL22650772

CC1(N)CCN(c2ccc(Nc3nccc(-c4cc(F)c5c(c4)C(C)(C)CO5)n3)nc2)C(=O)C1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 18/20 0.46
CCND3 P30281 8/20 0.46
CDK4 P11802 15/20 0.43
CCNA2 P20248 4/20 0.40
CDK1 P06493 3/20 0.40
CDK9 P50750 2/20 0.38
CCNT1 O60563 1/20 0.38
CCND1 P24385 1/20 0.38
CDK7 P50613 1/20 0.38
CCNH P51946 1/20 0.38
MNAT1 P51948 1/20 0.38
CDK5 Q00535 1/20 0.38
CDK5R1 Q15078 1/20 0.38
CDK2 P24941 3/20 0.37
PIK3CD O00329 3/20 0.37
CSF1R P07333 3/20 0.37
TYK2 P29597 2/20 0.37
CCNK O75909 1/20 0.37
CCNE2 O96020 1/20 0.37
PIM1 P11309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650771 0.93 CDK6 (0.43) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650492 0.86 CDK6 (0.58) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650509 0.84 CDK6 (0.48) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650773 0.83 CDK4 (0.45) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL29462408 0.81 DYRK2 (0.47) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650497 0.81 DYRK2 (0.47) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650507 0.80 CDK6 (0.45) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650755 0.74 CDK4 (0.42) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650705 0.74 CDK6 (0.39) CDK6CCND3CDK4CCNA2CDK1
SCHEMBL22650516 0.73 JAK2 (0.41) CDK6CCND3CDK4JAK2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed