SCHEMBL22650509

SCHEMBL22650509

CC1(C)COc2c(F)cc(-c3ccnc(Nc4ccc(N5CCCNC5=O)cn4)n3)cc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK6 Q00534 19/20 0.48
CCND3 P30281 10/20 0.48
CDK4 P11802 16/20 0.45
CCND1 P24385 5/20 0.45
CCNT1 O60563 2/20 0.45
CDK7 P50613 2/20 0.45
CDK9 P50750 2/20 0.45
CCNH P51946 2/20 0.45
MNAT1 P51948 2/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
CCNA2 P20248 6/20 0.44
CDK1 P06493 5/20 0.44
CDK2 P24941 5/20 0.42
CSF1R P07333 3/20 0.42
CCNE2 O96020 2/20 0.41
PIM1 P11309 2/20 0.41
PIK3CD O00329 2/20 0.40
CCNE1 P24864 1/20 0.39
CCNB1 P14635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22650492 0.87 CDK6 (0.58) CDK6CCND3CDK4CCND1CCNT1
SCHEMBL22650507 0.85 CDK6 (0.45) CDK6CCND3CDK4CCND1CDK7
SCHEMBL22650772 0.84 CDK6 (0.46) CDK6CCND3CDK4CCND1CCNT1
SCHEMBL22650773 0.82 CDK4 (0.45) CDK6CCND3CDK4CCND1CDK7
SCHEMBL29462408 0.79 DYRK2 (0.47) CDK6CCND3CDK4CCND1CCNT1
SCHEMBL22650497 0.79 DYRK2 (0.47) CDK6CCND3CDK4CCND1CCNT1
SCHEMBL22650771 0.79 CDK6 (0.43) CDK6CCND3CDK4CCND1CCNT1
SCHEMBL22650518 0.76 JAK2 (0.39) CDK6CCND3CDK4
SCHEMBL22650516 0.76 JAK2 (0.41) CDK6CCND3CDK4
SCHEMBL22650508 0.75 JAK2 (0.38) CDK6CCND3CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020224568-A1 CDK INHIBITORS QILU REGOR THERAPEUTICS INC. (CN) 2020-11-12 WO disclosed