Pentylenetetrazol

Pentylenetetrazol

SCHEMBL22674

C1CCc2nnnn2CC1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 1.00
MEN1 O00255 1/20 1.00
MAPT P10636 1/20 1.00
BLM P54132 1/20 1.00
KMT2A Q03164 1/20 1.00
POLB P06746 2/20 0.41
PDPK1 O15530 1/20 0.38
HPGD P15428 5/20 0.34
HTT P42858 2/20 0.33
RORC P51449 1/20 0.33
HSD11B1 P28845 3/20 0.33
HSD17B1 P14061 1/20 0.33
USP2 O75604 1/20 0.30
INMT O95050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pentylenetetrazol SCHEMBL6407957 1.00 ALDH1A1 (1.00) ALDH1A1MEN1MAPTBLMKMT2A
SCHEMBL3182039 1.00 ALDH1A1 (1.00) ALDH1A1MEN1MAPTBLMKMT2A
Pentylenetetrazol SCHEMBL9838533 1.00 ALDH1A1 (1.00) ALDH1A1MEN1MAPTBLMKMT2A
Pentylenetetrazol SCHEMBL10408117 0.98 ALDH1A1 (0.96) ALDH1A1MEN1MAPTBLMKMT2A
Pentylenetetrazol SCHEMBL15057132 0.98 ALDH1A1 (0.96) ALDH1A1MEN1MAPTBLMKMT2A
Pentylenetetrazol SCHEMBL10873243 0.98 ALDH1A1 (0.96) ALDH1A1MEN1MAPTBLMKMT2A
SCHEMBL2211329 0.98
SCHEMBL2212322 0.91
Pentylenetetrazol SCHEMBL2260235 0.87 ALDH1A1 (0.76) ALDH1A1MEN1MAPTBLMKMT2A
Biphenyl SCHEMBL7633644 0.86 ALDH1A1 (0.73) ALDH1A1MEN1MAPTBLMKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 15848 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4105216-B1 DIHYDRONAPHTHYRIDINONE COMPOUND, AND PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF GENFLEET THERAPEUTICS SHANGHAI INC (CN) 2026-05-20 EP claimed
EP-3986465-B1 SITE-SPECIFIC, KINETICALLY INERT CONJUGATION OF LABELS AND/OR CARRIERS TO TARGET MOLECULES SUCH AS HIS-TAGGED PROTEINS VIA METAL COMPLEX REAGENTS MAX PLANCK GESELLSCHAFT (DE) 2026-05-13 EP claimed
EP-4121423-B1 TETRAZOLE DERIVATIVES MERCK PATENT GMBH (DE) 2026-04-29 EP claimed
EP-4205191-B1 CHEMICAL COMPOUND, USE OF AT LEAST ONE SUCH CHEMICAL COMPOUND IN AN OPTOELECTRONIC COMPONENT, AND OPTOELECTRONIC COMPONENT CONTAINING AT LEAST ONE SUCH CHEMICAL COMPOUND HELIATEK GMBH (DE) 2026-04-22 EP claimed
EP-4722714-A1 SIMULTANEOUS ANALYSIS OF FOOD-BORNE DOPING SUBSTANCES USING LIQUID CHROMATOGRAPHY-MASS SPECTROMETRY (VFD: VACCINE FOR FOODBORNE DOPING) Korea Institute of Science and Technology (KR) 2026-04-08 EP claimed
EP-3768675-B1 NOVEL TRIAZOLONE DERIVATIVES OR SALTS THEREOF AND PHARMACEUTICAL COMPOSITIONS COMPRISING THE SAME YUHAN CORP (KR) 2026-04-01 EP claimed
EP-3995550-B1 POLISHING COMPOSITIONS AND METHODS OF USING SAME FUJIFILM ELECTRONIC MAT USA INC (US) 2026-04-01 EP claimed
EP-3820850-B1 PHENYL/PYRIDYL-N-PHENYL/PYRIDYL DERIVATIVES FOR TREATING A RNA VIRUS INFECTION ABIVAX (FR) 2026-04-01 EP claimed
EP-3723744-B1 C5AR INHIBITORS FOR USE IN THE TREATMENT OF CHEMOTHERAPY-INDUCED IATROGENIC PAIN DOMPE FARM SPA (IT) 2026-03-18 EP claimed
US-20260062760-A1 METHODS OF TREATMENT AND DIAGNOSIS OF MULTIPLE MYELOMA PROGRESSION MOREHOUSE SCHOOL OF MEDICINE (US) 2026-03-05 US claimed
EP-0034925-B1 5-(DIHYDROXYPHENOXY) TETRAZOLES AS SWEETENERS ELI LILLY AND COMPANY (US) 1983-05-04 EP claimed
EP-0000500-B1 CEPHALOSPRIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM CIBA-GEIGY AG (CH) 1982-04-28 EP claimed
EP-0004570-B1 THIOL ESTERS, PROCESS FOR THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND A PROCESS FOR PREPARING CEPHALOSPORIN COMPOUNDS USING THE SAME Asahi Kasei Kogyo Kabushiki Kaisha (JP) 1982-04-14 EP claimed
EP-0002586-B1 METHOD FOR REMOVING A HALOGENOACETYL PROTECTIVE GROUP FROM A HALOGENOACETYL AMINO COMPOUND Takeda Chemical Industries, Ltd. (JP) 1982-01-20 EP claimed
EP-0035046-A1 Novel tetrazole derivatives, process for the preparation thereof, and anti-ulcer composition containing the same OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1981-09-09 EP claimed
US-4243748-A DIHETEROCYCLIC DISULFIDE, THIAZOLIDINECARBOXYLIC COMPOUND E. I. DU PONT DE NEMOURS AND COMPANY (US) 1981-01-06 US claimed
EP-0011092-A1 Alpha-aminophenylacetic acid derivatives for use in the treatment of inflammations and novel alpha-aminophenylacetic acid derivatives BAYER AG (DE) 1980-05-28 EP claimed
US-4187221-A Process for preparing azetidinones CONNLAB HOLDINGS LIMITED (CA) 1980-02-05 US claimed
US-4045306-A REACTION PRODUCT OF UNSATURATED NITROGEN HETEROCYCLIC COMPOUND AND A HALOHYDRIN SCHERING AKTIENGESELLSCHAFT (DT) 1977-08-30 US claimed
US-3989696-A 3-Heterothio[(oxyalkyl)thioacetyl]cephalosporin derivatives E. R. SQUIBB & SONS, INC. (US) 1976-11-02 US claimed